Optimization of permeability in a series of pyrrolotriazine inhibitors of IRAK4

Bibliographic Details
Title: Optimization of permeability in a series of pyrrolotriazine inhibitors of IRAK4
Authors: Degorce, Sébastien L., Anjum, Rana, Dillman, Keith S., Drew, Lisa, Groombridge, Sam D., Halsall, Christopher T., Lenz, Eva M., Lindsay, Nicola A., Mayo, Michele F., Pink, Jennifer H., Robb, Graeme R., Scott, James S., Stokes, Stephen, Xue, Yafeng
Source: In Bioorganic & Medicinal Chemistry 15 February 2018 26(4):913-924
Database: ScienceDirect
More Details
ISSN:09680896
DOI:10.1016/j.bmc.2018.01.008
Published in:Bioorganic & Medicinal Chemistry
Language:English