Identification of novel series of pyrazole and indole-urea based DFG-out PYK2 inhibitors

Bibliographic Details
Title: Identification of novel series of pyrazole and indole-urea based DFG-out PYK2 inhibitors
Authors: Bhattacharya, Samit K., Aspnes, Gary E., Bagley, Scott W., Boehm, Markus, Brosius, Arthur D., Buckbinder, Leonard, Chang, Jeanne S., Dibrino, Joseph, Eng, Heather, Frederick, Kosea S., Griffith, David A., Griffor, Matthew C., GuimarĂ£es, Cristiano R.W., Guzman-Perez, Angel, Han, Seungil, Kalgutkar, Amit S., Klug-McLeod, Jacquelyn, Garcia-Irizarry, Carmen, Li, Jianke, Lippa, Blaise, Price, David A., Southers, James A., Walker, Daniel P., Wei, Liuqing, Xiao, Jun, Zawistoski, Michael P., Zhao, Xumiao
Source: In Bioorganic & Medicinal Chemistry Letters 15 December 2012 22(24):7523-7529
Database: ScienceDirect
More Details
ISSN:0960894X
DOI:10.1016/j.bmcl.2012.10.039
Published in:Bioorganic & Medicinal Chemistry Letters
Language:English