Discovery of 22(S)-23-phenyl-24-norchol-5-en-3β,22-diol (PFM046) as the first-in-class, steroidal, non-sulfated Liver X Receptor antagonist with anticancer activity

Bibliographic Details
Title: Discovery of 22(S)-23-phenyl-24-norchol-5-en-3β,22-diol (PFM046) as the first-in-class, steroidal, non-sulfated Liver X Receptor antagonist with anticancer activity
Authors: Pontini, Lorenzo a, 1, Angelini, Tommaso a, 1, Palazzoli, Pietro a, 1, Maggioni, Daniela b, Giorgi, Gianluca c, Raccosta, Laura b, Damiano, Giuseppe b, Mammoli, Valerio d, Fontana, Niccolò d, Russo, Vincenzo b, ⁎⁎, Marinozzi, Maura a, ⁎
Source: In European Journal of Medicinal Chemistry 5 February 2025 283
Database: ScienceDirect
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ISSN:02235234
DOI:10.1016/j.ejmech.2024.117136
Published in:European Journal of Medicinal Chemistry
Language:English