A Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug Discovery
Title: | A Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug Discovery |
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Authors: | Hafey, Michael J. *, Houle, Robert, Tanis, Keith Q., Knemeyer, Ian, Shang, Jackie 1, Chen, Qing 2, Baudy, Andreas, Monroe, James, Sistare, Frank D., Evers, Raymond 3 |
Source: | In Drug Metabolism and Disposition November 2020 48(11):1147-1160 |
Database: | ScienceDirect |
ISSN: | 00909556 |
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DOI: | 10.1124/dmd.120.000086 |
Published in: | Drug Metabolism and Disposition |
Language: | English |