A Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug Discovery

Bibliographic Details
Title: A Two-Tiered In Vitro Approach to De-Risk Drug Candidates for Potential Bile Salt Export Pump Inhibition Liabilities in Drug Discovery
Authors: Hafey, Michael J. *, Houle, Robert, Tanis, Keith Q., Knemeyer, Ian, Shang, Jackie 1, Chen, Qing 2, Baudy, Andreas, Monroe, James, Sistare, Frank D., Evers, Raymond 3
Source: In Drug Metabolism and Disposition November 2020 48(11):1147-1160
Database: ScienceDirect
More Details
ISSN:00909556
DOI:10.1124/dmd.120.000086
Published in:Drug Metabolism and Disposition
Language:English