Slow-, Tight-Binding Inhibition of CYP17A1 by Abiraterone Redefines Its Kinetic Selectivity and Dosing Regimen

Bibliographic Details
Title: Slow-, Tight-Binding Inhibition of CYP17A1 by Abiraterone Redefines Its Kinetic Selectivity and Dosing Regimen
Authors: Cheong, Eleanor Jing Yi, Nair, Pramod C., Neo, Rebecca Wan Yi, Tu, Ho Thanh, Lin, Fu, Chiong, Edmund, Esuvaranathan, Kesavan, Fan, Hao, Szmulewitz, Russell Z., Peer, Cody J., Figg, William D., Chai, Christina Li Lin, Miners, John O., Chan, Eric Chun Yong *
Source: In The Journal of Pharmacology and Experimental Therapeutics September 2020 374(3):438-451
Database: ScienceDirect
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ISSN:00223565
DOI:10.1124/jpet.120.265868
Published in:The Journal of Pharmacology and Experimental Therapeutics
Language:English