Structural and Biochemical Analyses Reveal the Mechanism of Glutathione S-Transferase Pi 1 Inhibition by the Anti-cancer Compound Piperlongumine

Bibliographic Details
Title: Structural and Biochemical Analyses Reveal the Mechanism of Glutathione S-Transferase Pi 1 Inhibition by the Anti-cancer Compound Piperlongumine
Alternate Title: Hydrolyzed Piperlongumine Inhibits GSTP1 (English)
Authors: Harshbarger, Wayne, Gondi, Sudershan, Ficarro, Scott B., Hunter, John, Udayakumar, Durga, Gurbani, Deepak, Singer, William D., Liu, Yan, Li, Lianbo, Marto, Jarrod A., Westover, Kenneth D.
Source: In Journal of Biological Chemistry 6 January 2017 292(1):112-120
Database: ScienceDirect
More Details
ISSN:00219258
DOI:10.1074/jbc.M116.750299
Published in:Journal of Biological Chemistry
Language:English