Why Is Quinidine an Inhibitor of Cytochrome P450 2D6?: THE ROLE OF KEY ACTIVE-SITE RESIDUES IN QUINIDINE BINDING
Title: | Why Is Quinidine an Inhibitor of Cytochrome P450 2D6?: THE ROLE OF KEY ACTIVE-SITE RESIDUES IN QUINIDINE BINDING |
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Authors: | McLaughlin, Lesley A. ‡, 1, Paine, Mark J.I. ‡, 1, Kemp, Carol A. §, Maréchal, Jean-Didier §, ¶, Flanagan, Jack U. ‡, Ward, Clive J. ‡, Sutcliffe, Michael J. §, ¶, Roberts, Gordon C.K. §, 2, Wolf, C. Roland ‡, 3 |
Source: | In Journal of Biological Chemistry 18 November 2005 280(46):38617-38624 |
Database: | ScienceDirect |
ISSN: | 00219258 |
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DOI: | 10.1074/jbc.M505974200 |
Published in: | Journal of Biological Chemistry |
Language: | English |