Illuminating the Dark: Highly Selective Inhibition of Serine/Threonine Kinase 17A with Pyrazolo[1,5‑a]pyrimidine-Based Macrocycles.

Bibliographic Details
Title: Illuminating the Dark: Highly Selective Inhibition of Serine/Threonine Kinase 17A with Pyrazolo[1,5‑a]pyrimidine-Based Macrocycles.
Authors: Kurz, Christian G.1,2 (AUTHOR), Preuss, Franziska1,2 (AUTHOR), Tjaden, Amelie1,2 (AUTHOR), Cusack, Martin3 (AUTHOR), Amrhein, Jennifer Alisa1,2 (AUTHOR), Chatterjee, Deep1,2 (AUTHOR), Mathea, Sebastian1,2 (AUTHOR), Berger, Lena Marie1,2 (AUTHOR), Berger, Benedict-Tilman1,2 (AUTHOR), Krämer, Andreas1,2,4 (AUTHOR), Weller, Michael3 (AUTHOR), Weiss, Tobias3 (AUTHOR), Müller, Susanne1,2 (AUTHOR), Knapp, Stefan1,2 (AUTHOR) knapp@pharmchem.uni-frankfurt.de, Hanke, Thomas1,2 (AUTHOR) hanke@pharmchem.uni-frankfurt.de
Source: Journal of Medicinal Chemistry. 6/9/2022, Vol. 65 Issue 11, p7799-7817. 19p.
Database: Supplemental Index
More Details
ISSN:00222623
DOI:10.1021/acs.jmedchem.2c00173
Published in:Journal of Medicinal Chemistry
Language:English