Discovery of a Potent and Selective ATAD2 Bromodomain Inhibitor with Antiproliferative Activity in Breast Cancer Models.

Bibliographic Details
Title: Discovery of a Potent and Selective ATAD2 Bromodomain Inhibitor with Antiproliferative Activity in Breast Cancer Models.
Authors: Winter-Holt, Jon J., Bardelle, Catherine, Chiarparin, Elisabetta, Dale, Ian L., Davey, Paul R. J., Davies, Nichola L., Denz, Christopher, Fillery, Shaun M., Guérot, Carine M., Fujin Han, Hughes, Samantha J., Kulkarni, Meghana, Zhaoqun Liu, Milbradt, Alexander, Moss, Thomas A., Huijun Niu, Patel, Joe, Rabow, Alfred A., Schimpl, Marianne, Junjie Shi
Source: Journal of Medicinal Chemistry; 2/24/2022, Vol. 65 Issue 4, p3306-3331, 26p
Database: Supplemental Index
More Details
ISSN:00222623
DOI:10.1021/acs.jmedchem.1c01871
Published in:Journal of Medicinal Chemistry
Language:English