Rational Design and Optimization of a Novel Class of Macrocyclic Apoptosis Signal-Regulating Kinase 1 Inhibitors.

Bibliographic Details
Title: Rational Design and Optimization of a Novel Class of Macrocyclic Apoptosis Signal-Regulating Kinase 1 Inhibitors.
Authors: Himmelbauer, Martin K., Xin, Zhili, Jones, J. Howard, Enyedy, Istvan, King, Kristopher, Marcotte, Douglas J., Murugan, Paramasivam, Santoro, Joseph C., Hesson, Thomas, Spilker, Kerri, Johnson, Joshua L., Luzzio, Michael J., Gilfillan, Rab, de Turiso, Felix Gonzalez-Lopez
Source: Journal of Medicinal Chemistry; 12/12/2019, Vol. 62 Issue 23, p10740-10756, 17p
Database: Supplemental Index
More Details
ISSN:00222623
DOI:10.1021/acs.jmedchem.9b01206
Published in:Journal of Medicinal Chemistry
Language:English