Heterotropic allosteric modulation of CYP3A4 in vitro by progesterone: Evidence for improvement in prediction of time-dependent inhibition for macrolides
Title: | Heterotropic allosteric modulation of CYP3A4 in vitro by progesterone: Evidence for improvement in prediction of time-dependent inhibition for macrolides |
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Authors: | Rougée, Luc R.A. ∗, Hegde, Pooja V., Shin, Kaitlin, Abraham, Trent L., Bell, Alec, Hall, Stephen D. |
Source: | In Drug Metabolism and Disposition January 2025 53(1) |
Database: | ScienceDirect |
ISSN: | 00909556 |
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DOI: | 10.1124/dmd.124.001820 |
Published in: | Drug Metabolism and Disposition |
Language: | English |