A First-in-Class Pyrazole-isoxazole Enhanced Antifungal Activity of Voriconazole: Synergy Studies in an Azole-Resistant Candida albicans Strain, Computational Investigation and in Vivo Validation in a Galleria mellonella Fungal Infection Model.

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Title: A First-in-Class Pyrazole-isoxazole Enhanced Antifungal Activity of Voriconazole: Synergy Studies in an Azole-Resistant Candida albicans Strain, Computational Investigation and in Vivo Validation in a Galleria mellonella Fungal Infection Model.
Authors: Pelliccia, Sveva, Russomanno, Pasquale, Barone, Simona, Mateu, Baptiste, Alfano, Antonella Ilenia, Miranda, Martina, Coretti, Lorena, Lembo, Francesca, Piccolo, Marialuisa, Irace, Carlo, Friggeri, Laura, Hargrove, Tatiana Y., Curtis, Aaron, Lepesheva, Galina I., Kavanagh, Kevin, Buommino, Elisabetta, Brindisi, Margherita
Source: Journal of Medicinal Chemistry; 8/22/2024, Vol. 671 Issue 6, p14256-14276, 21p
Database: Supplemental Index
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  Data: Journal of Medicinal Chemistry; 8/22/2024, Vol. 671 Issue 6, p14256-14276, 21p
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        Value: 10.1021/acs.jmedchem.4c01109
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      – TitleFull: A First-in-Class Pyrazole-isoxazole Enhanced Antifungal Activity of Voriconazole: Synergy Studies in an Azole-Resistant Candida albicans Strain, Computational Investigation and in Vivo Validation in a Galleria mellonella Fungal Infection Model.
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              Text: 8/22/2024
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