Control of Neurotransmission by NaV1.7 in Human, Guinea Pig, and Mouse Airway Parasympathetic Nerves

Authors: Kocmalova, Michaela, Kollarik, Marian, Canning, Brendan. J., Ru, Fei, Adam Herbstsomer, R., Meeker, Sonya, Fonquerna, Silvia, Aparici, Monica, Miralpeix, Montserrat, Chi, Xian Xuan, Li, Baolin, Wilenkin, Ben, McDermott, Jeff, Nisenbaum, Eric, Krajewski, Jeffrey L., Undem, Bradley J. ^*

Source: In The Journal of Pharmacology and Experimental Therapeutics April 2017 361(1):172-180

The discovery of aminopyrazines as novel, potent Nav1.7 antagonists: Hit-to-lead identification and SAR

Authors: Bregman, Howard, Nguyen, Hanh Nho, Feric, Elma, Ligutti, Joseph, Liu, Dong, McDermott, Jeff S., Wilenkin, Ben, Zou, Anruo, Huang, Liyue, Li, Xingwen, McDonough, Stefan I., DiMauro, Erin F.

Source: In Bioorganic & Medicinal Chemistry Letters 1 March 2012 22(5):2033-2042

Discovery and optimization of aminopyrimidinones as potent and state-dependent Nav1.7 antagonists

Authors: Nguyen, Hanh Nho, Bregman, Howie, Buchanan, John L., Du, Bingfan, Feric, Elma, Huang, Liyue, Li, Xingwen, Ligutti, Joseph, Liu, Dong, Malmberg, Annika B., Matson, David J., McDermott, Jeff S., Patel, Vinod F., Wilenkin, Ben, Zou, Anruo, McDonough, Stefan I., DiMauro, Erin F.

Source: In Bioorganic & Medicinal Chemistry Letters 15 January 2012 22(2):1055-1060

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