Convergent synthesis of dihydroquinolones from o-aminoarylboronates
Modern applications of transition metal catalysis in heterocycle synthesis: tetrahedron symposium in print number 146

Authors: Horn, J., Li, H. Y., Marsden, S. P., Nelson, A., Shearer, R. J., Campbell, A. J., House, D., Weingarten, G. G.

Source: TETRAHEDRON -LONDON-. 65(44):9002-9007

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCCN074273553&indx=1&recIds=ETOCCN074273553

Synthesis and in vivo biological activity of large-ringed calixarenes against Mycobacterium tuberculosis

Authors: Goodworth, K. J., Herve, A. C., Stavropoulos, E., Herve, G., Casades, I., Hill, A. M., Weingarten, G. G., Tascon, R. E., Colston, M. J., Hailes, H. C.

Source: TETRAHEDRON -LONDON-. 67(2):373-382

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Design and Synthesis of Pyrrolidine-5,5-trans-lactams as Novel Mechanism Based Inhibitors of Human Cytomegalovirus Protease

Authors: Borthwick, A. D., Crame, A. J., Ertl, P. F., Exall, A. M., Haley, T. M., Hart, G. J., Mason, A. M., Pennell, A. M. K., Singh, O. M. P., Weingarten, G. G.

Source: CHEMTRACTS -NEW YORK-. 15(7):367-372

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Pyrrolidine-5,5-trans-lactams as novel mechanism-based inhibitors of human cytomegalovirus protease. Part 3: potency and plasma stability

Authors: Borthwick, A. D., Exall, A. M., Haley, T. M., Jackson, D. L., Mason, A. M., Weingarten, G. G.

Source: BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS. 12(13):1719-1722

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Identification of potent and selective oxytocin antagonists. Part 2: further investigation of benzofuran derivatives

Authors: Wyatt, P. G., Allen, M. J., Chilcott, J., Gardner, C. J., Livermore, D. G., Mordaunt, J. E., Nerozzi, F., Patel, M., Perren, M. J., Weingarten, G. G.

Source: BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS. 12(10):1405-1411

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Design and Synthesis of Pyrrolidine-5,5-trans-lactams (5-Oxohexahydropyrrolo[3,2-b]pyrroles) as Novel Mechanism-Based Inhibitors of Human Cytomegalovirus Protease. 2. Potency and Chirality

Authors: Borthwick, A. D., Crame, A. J., Ertl, P. F., Exall, A. M., Haley, T. M., Hart, G. J., Mason, A. M., Pennell, A. M. K., Singh, O. M. P., Weingarten, G. G.

Source: JOURNAL OF MEDICINAL CHEMISTRY. 45(1):1-18

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Design and Synthesis of Pyrrolidine-5,5-trans-lactams (5-Oxo-hexahydro-pyrrolo[3,2-b]pyrroles) as Novel Mechanism-Based Inhibitors of Human Cytomegalovirus Protease. 1. The alpha-Methyl-trans-lactam Template

Authors: Borthwick, A. D., Angier, S. J., Crame, A. J., Exall, A. M., Haley, T. M., Hart, G. J., Mason, A. M., Pennell, A. M. K., Weingarten, G. G.

Source: JOURNAL OF MEDICINAL CHEMISTRY. 43(23):4452-4464

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A study of the stereochemical features of 5-endo-trig iodocyclisations of 2-alkenylcycloalkan-1-ols

Authors: Barks, J. M., Weingarten, G. G., Knight, D. W.

Source: PERKIN 1. (20):3469-3476

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Stereoselective Synthesis of alpha-Methyl and beta-Methyl Pyrrolidine 5,5-trans-Lactam (5-Oxo-hexahydropyrrolo[3,2-b]pyrrole) and Stereoselective Alkylation of the Strained Pyrrolidine 5,5-Trans-Lactam Ring System

Authors: Borthwick, A. D., Crame, A. J., Davies, D. E., Exall, A. M., Jackson, D. L., Mason, A. M., Pennell, A. M., Weingarten, G. G.

Source: SYNLETT. (4):504-508

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An efficient synthesis of a chiral carbocyclic 2'-deoxyribonucleoside synthon by directed reduction

Authors: Borthwick, A. D., Crame, A. J., Exall, A. M., Weingarten, G. G.

Source: TETRAHEDRON LETTERS. 35(41):7677-7677

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Predictive models for the overall 5-endo-trig iodocyclisation of homoallylic alcohols

Authors: Barks, J. M., Knight, D. W., Seaman, C. J., Weingarten, G. G.

Source: TETRAHEDRON LETTERS. 35(39):7259-7259

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCEN020229469&indx=1&recIds=ETOCEN020229469

Pyrrolidine-5,5-Translactams, Novel Herpes Protease Inhibitors that are Potent Antivirals Against Human Cytomegalovirus

Authors: Borthwick, A. D., Crame, A., Exall, A. M., Jackson, D. L., Mason, A. M., Pennell, A. M. K., Weingarten, G. G., Haley, T. M., Hart, G. J., Parry, N. R.

Source: ANTIVIRAL RESEARCH. 41(2):14-14

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A Short High Yielding Synthesis of the Potent Anti-VZV Carbocyclic Nucleoside Analogue Carba-BVDU.

Authors: Wyatt, P. G., Anslow, A. S., Coomber, B. A., Cousins, R. P.C., Evans, D. N., Gilbert, V. S., Humber, D. C., Paternoster, I. L., Sollis, S. L., Tapolczay, D. J., Weingarten, G. G.

Source: Nucleosides & Nucleotides; Nov1995, Vol. 14 Issue 9/10, p2039-2049, 11p

Photochemical transformations. Part XXVIII. Aryl azides as potential photosensitive protecting groups.

Authors: Barton, D. H. R., Sammes, P. G., Weingarten, G. G.

Source: Journal of the Chemical Society C: Organic; 1971, p721-728, 8p

Photochemical transformations. Part XXIX. Steric compression effects in the synthesis and reactions of 4-amino-5-methylphenanthrene.

Authors: Barton, D. H. R., Sammes, P. G., Weingarten, G. G.

Source: Journal of the Chemical Society C: Organic; 1971, p729-736, 8p

Design and Synthesis of Pyrrolidine-5,5‘-trans-Lactams (5-Oxo-hexahydropyrrolo[3,2-b]pyrroles) as Novel Mechanism-Based Inhibitors of Human Cytomegalovirus Protease. 4. Antiviral Activity and Plasma Stability

Authors: Borthwick, A. D., Davies, D. E., Ertl, P. F., Exall, A. M., Haley, T. M., Hart, G. J., Jackson, D. L., Parry, N. R., Patikis, A., Trivedi, N., Weingarten, G. G., Woolven, J. M.

Source: Journal of Medicinal Chemistry; October 2003, Vol. 46 Issue: 21 p4428-4449, 22p

Design and Synthesis of Pyrrolidine-5,5-trans-lactams (5-Oxo-hexahydro-pyrrolo[3,2-b]pyrroles) as Novel Mechanism-Based Inhibitors of Human Cytomegalovirus Protease. 1. The α-Methyl-trans-lactam Template

Authors: Borthwick, A. D., Angier, S. J., Crame, A. J., Exall, A. M., Haley, T. M., Hart, G. J., Mason, A. M., Pennell, A. M. K., Weingarten, G. G.

Source: Journal of Medicinal Chemistry; November 16, 2000, Vol. 43 Issue: 23 p4452-4464, 13p

Synthesis and Structure Activity Relationships of a Series of Penicillin-Derived Pseudosymmetric Inhibitors of HIV-1 Proteinase

Authors: Humber, D. C., Bamford, M. J., Bethell, R. C., Cammack, N., Orr, D. C., Storer, R., Weingarten, G. G., Wyatt, P. G.

Source: Antiviral Chemistry & Chemotherapy; June 1994, Vol. 5 Issue: 3 p197-200, 4p

Improved Synthesis of (−)-Carbovir, GR90352X, a Potent and Selective Inhibitor of HIV-1 in Vitro.

Authors: JONES, M. F., MO, C. L., MYERS, P. L., PATERNOSTER, I. L., STORER, R., WEINGARTEN, G. G., WILLIAMSON, C.

Source: Annals of the New York Academy of Sciences; 1991, Vol. 616 Issue 1, p535-537, 3p

ChemInform Abstract: A Short High Yielding Synthesis of the Potent anti-VZV Carbocyclic Nucleoside Analogue Carba-BVDU.

Authors: WYATT, P. G., ANSLOW, A. S., COOMBER, B. A., COUSINS, R. P. C., EVANS, D. N., GILBERT, V. S., HUMBER, D. C., PATERNOSTER, I. L., SOLLIS, S. L., TAPOLCZAY, D. J., WEINGARTEN, G. G.

Source: ChemInform; Apr1996, Vol. 27 Issue 16, pno-no, 1p