One-step hydroxylation of aryl and heteroaryl fluorides using mechanochemistryElectronic supplementary information (ESI) available. See DOI: 10.1039/d1gc04361g

Authors: Rodrigo, Eduardo, Wiechert, Rainer, Walter, Magnus W., Braje, Wilfried, Geneste, Hervé

Source: Green chemistry. 24(4):1469-1473

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100141638067.0x000001&indx=1&recIds=ETOCvdc_100141638067.0x000001

A pharma-wide approach to address the genotoxicity prediction of primary aromatic amines

Authors: Patel, Mukesh, Kranz, Michael, Munoz-Muriedas, Jordi, Harvey, James S., Giddings, Amanda, Swallow, Steve, Fellows, Mick, Naven, Russell, Werner, Anne-Laure, Yeo, David J., Bringezu, Frank, Wichard, Joerg, Sutter, Andreas, Glowienke, Susanne, Whitehead, Lewis, Selby, Matt, Reuberson, James, Atienzar, Franck, Gerets, Helga, Kenyon, Michelle O., Dobo, Krista L., Walter, Magnus W., Jolly, Robert A., Amberg, Alexander, Spirkl, Hans-Peter, Muster, Wolfgang, Van Gompel, Jacques

Source: In Computational Toxicology August 2018 7:27-35

Neurochemical and behavioral profiling of the selective GlyT1 inhibitors ALX5407 and LY2365109 indicate a preferential action in caudal vs. cortical brain areas

Authors: Perry, Kenneth W., Falcone, Julie F., Fell, Matthew J., Ryder, John W., Yu, Hong, Love, Patrick L., Katner, Jason, Gordon, Kimberly D., Wade, Mark R., Man, Teresa, Nomikos, George G., Phebus, Lee A., Cauvin, Annick J., Johnson, Kirk W., Jones, Carrie K., Hoffmann, Beth J., Sandusky, George E., Walter, Magnus W., Porter, Warren J., Yang, Lijuan, Merchant, Kalpana M., Shannon, Harlan E., Svensson, Kjell A.

Source: In Neuropharmacology 2008 55(5):743-754

Synthesis of 11C-labelled ( R)-OHDMI and CFMME and their evaluation as candidate radioligands for imaging central norepinephrine transporters with PET

Authors: Schou, Magnus, Pike, Victor W., Sóvágó, Judit, Gulyás, Balázs, Gallagher, Peter T., Dobson, David R., Walter, Magnus W., Rudyk, Helene, Farde, Lars, Halldin, Christer

Source: In Bioorganic & Medicinal Chemistry 2007 15(2):616-625

Total synthesis of cyercene A and the biomimetic synthesis of (±)-9,10-deoxytridachione and (±)-ocellapyrone A

Authors: Rodriguez, Raphaël, Adlington, Robert M., Eade, Serena J., Walter, Magnus W., Baldwin, Jack E., Moses, John E.

Source: In Tetrahedron 2007 63(21):4500-4509

Biomimetic Synthesis of Pyrone-Derived Natural Products: Exploring Chemical Pathways from a Unique Polyketide Precursor.

Authors: Eade, Serena J., Walter, Magnus W., Byrne, Colin

Source: Journal of Organic Chemistry; July 4 2008, Vol. 73 Issue 13, p4830-4839, 10p

Perfluoralkyl substituted metallo-beta-lactamase inhibitors

Reaction of (trifluoromethyl)trimethylsilane with oxazolidin-5-ones: synthesis of peptidic and nonpeptidic trifluoromethyl ketones.

Authors: Walter, Magnus W., Adlington, Robert M., Baldwin, Jack E.

Source: Journal of Organic Chemistry; July 24 1998, Vol. 63 Issue 15, p5179-5192, 14p

Screening of a Custom-Designed Acid Fragment Library Identifies 1‑Phenylpyrroles and 1‑Phenylpyrrolidines as Inhibitors of Notum Carboxylesterase Activity.

Authors: Mahy, William, Patel, Mikesh, Steadman, David, Woodward, Hannah L., Atkinson, Benjamin N., Svensson, Fredrik, Willis, Nicky J., Flint, Alister, Papatheodorou, Dimitra, Zhao, Yuguang, Vecchia, Luca, Ruza, Reinis R., Hillier, James, Frew, Sarah, Monaghan, Amy, Costa, Artur, Bictash, Magda, Walter, Magnus W., Jones, E. Yvonne, Fish, Paul V.

Source: Journal of Medicinal Chemistry; 9/10/2020, Vol. 63 Issue 17, p9464-9483, 20p

Hydroxamate Inhibitors ofAeromonas hydrophilaAE036 Metallo-B-lactamase

Authors: Walter, Magnus W., Valladares, Maria Hernandez, Adlington, Robert M., Amicosante, Gianfranco, Baldwin, Jack E., Frère, Jean-Marie, Galleni, Moreno, Rossolini, Gian Maria, Schofield, Christopher J. ¹

Source: In Bioorganic Chemistry February 1999 27(1):35-40

This result is not displayed to guests.
Login for full access.

This result is not displayed to guests.
Login for full access.

Discovery and SAR studies of novel GlyT1 inhibitors

Authors: Walter, Magnus W., Hoffman, Beth J., Gordon, Kimberly, Johnson, Kirk, Love, Patrick, Jones, Matthew, Man, Teresa, Phebus, Lee, Reel, Jon K., Rudyk, Helene C., Shannon, Harlan, Svensson, Kjell, Yu, Hong, Valli, Matthew J., Porter, Warren J.

Source: In Bioorganic & Medicinal Chemistry Letters 2007 17(18):5233-5238

Discovery of novel and selective tertiary alcohol containing inhibitors of the norepinephrine transporter

Authors: Cases-Thomas, Manuel J., Masters, John J., Walter, Magnus W., Campbell, Gordon, Haughton, Louise, Gallagher, Peter T., Dobson, David R., Mancuso, Vincent, Bonnier, Benjamin, Giard, Thierry, Defrance, Thierry, Vanmarsenille, Michel, Ledgard, Andrew, White, Craig, Ouwerkerk-Mahadevan, Sivi, Brunelle, Francoise J., Dezutter, Nancy A., Herbots, Camy A., Lienard, Joel Y., Findlay, Jeremy, Hayhurst, Lorna, Boot, John, Thompson, Linda K., Hemrick-Luecke, Susan

Source: In Bioorganic & Medicinal Chemistry Letters 2006 16(7):2022-2025

1-Aryl-3,4-dihydro-1 H-quinolin-2-one derivatives, novel and selective norepinephrine reuptake inhibitors

Authors: Beadle, Christopher D., Boot, John, Camp, Nicholas P., Dezutter, Nancy, Findlay, Jeremy, Hayhurst, Lorna, Masters, John J., Penariol, Roberta, Walter, Magnus W.

Source: In Bioorganic & Medicinal Chemistry Letters 2005 15(20):4432-4437

Discovery and structure–activity relationships of novel selective norepinephrine and dual serotonin/norepinephrine reuptake inhibitors

Authors: Boot, John, Cases, Manuel, Clark, Barry P., Findlay, Jeremy, Gallagher, Peter T., Hayhurst, Lorna, Man, Teresa, Montalbetti, Christian, Rathmell, Richard E., Rudyk, Hélène, Walter, Magnus W. ^*, Whatton, Maria, Wood, Virginia

Source: In Bioorganic & Medicinal Chemistry Letters 2005 15(3):699-703

Monoamine reuptake inhibitors: highlights of recent research developments

Authors: Walter, Magnus W.

Source: Drug Development Research; July 2005, Vol. 65 Issue: 3 p97-118, 22p

Structure-based design of agrochemicals

Authors: Walter, Magnus W.

Source: Natural Product Reports; May 23, 2002, Vol. 19 Issue: 3 p278-291, 14p

Reaction of ruppert’s reagent (TMS-CF3) with Oxazolidinones: Synthesis of protected α-amino trifluoromethylketones

Authors: Walter, Magnus W., Adlington, Robert M., Baldwin, Jack E., Chuhan, John, Schofield, Christopher J.

Source: Tetrahedron Letters; October 1995, Vol. 36 Issue: 42 p7761-7764, 4p

This result is not displayed to guests.
Login for full access.