Purine containing carbonucleoside phosphonate analogues as novel chemotype for Plasmodium falciparum Inhibition

Authors: Mohamed, Bemba Sidi, Nguyen, Minh Chau, Wein, Sharon, Uttaro, Jean-Pierre, Robert, Xavier, Violot, Sébastien, Ballut, Lionel, Jugnarain, Vinesh, Mathé, Christophe, Cerdan, Rachel, Aghajari, Nushin, Peyrottes, Suzanne

Source: In European Journal of Medicinal Chemistry 5 October 2023 258

Third‐Generation CD73 Inhibitors Based on a 4,6‐Disubstituted‐2‐Thiopyridine Scaffold.

Authors: Grosjean, Félix, Shaldaeva, Maria, Cros‐Perrial, Emeline, Rodriguez, Céline, Ghoteimi, Rayane, Lebrun, Aurélien, Gao, Zhan‐Guo, Uttaro, Jean‐Pierre, Mathé, Christophe, Jacobson, Kenneth A., Petter Jordheim, Lars, Ménétrier‐Caux, Christine, Chaloin, Laurent, Peyrottes, Suzanne

Source: ChemMedChem; 3/15/2025, Vol. 20 Issue 6, p1-24, 24p

4-Substituted-1,2,3-triazolo nucleotide analogues as CD73 inhibitors, their synthesis, in vitro screening, kinetic and in silico studies

Authors: Ghoteimi, Rayane, Braka, Abdennour, Rodriguez, Céline, Cros-Perrial, Emeline, Tai Nguyen, Van, Uttaro, Jean-Pierre, Mathé, Christophe, Chaloin, Laurent, Ménétrier-Caux, Christine, Jordheim, Lars Petter, Peyrottes, Suzanne

Source: In Bioorganic Chemistry February 2021 107

Synthesis of 3′-halo-5′-norcarbocyclic nucleoside phosphonates as potent anti-HIV agents

Authors: Hamon, Nadège, Kaci, Malika, Uttaro, Jean-Pierre, Périgaud, Christian, Mathé, Christophe

Source: In European Journal of Medicinal Chemistry 25 April 2018 150:642-654

Synthesis of novel 3′-methyl-5′-norcarbocyclic nucleoside phosphonates as potential anti-HIV agents

Authors: Uttaro, Jean-Pierre, Broussous, Sylvie, Mathé, Christophe, Périgaud, Christian

Source: In Tetrahedron 4 March 2013 69(9):2131-2136

Synthesis of the natural enantiomer of neplanocin B

Authors: Hamon, Nadège, Uttaro, Jean-Pierre, Mathé, Christophe, Périgaud, Christian

Source: In Bioorganic Chemistry 2010 38(6):275-278

Second‐Generation CD73 Inhibitors Based on a 4,6‐Biaryl‐2‐thiopyridine Scaffold.

Authors: Ghoteimi, Rayane, Braka, Abdennour, Rodriguez, Céline, Cros‐Perrial, Emeline, Duvauchelle, Valentin, Uttaro, Jean‐Pierre, Mathé, Christophe, Ménétrier‐Caux, Christine, Jordheim, Lars Petter, Chaloin, Laurent, Peyrottes, Suzanne

Source: ChemMedChem; 4/3/2023, Vol. 18 Issue 7, p1-16, 16p

Discovery of an L‐like Configuration for 3'‐Fluoro‐5'‐norcarbonucleoside Phosphonates as Potent Anti‐HIV Agents.

Authors: Geant, Pierre‐Yves, Kaci, Malika, Uttaro, Jean‐Pierre, Périgaud, Christian, Mathé, Christophe

Source: ChemMedChem; 10/19/2022, Vol. 17 Issue 20, p1-8, 8p

Chemoenzymatic Taxanes Approach Using Both Enantiomers of the Same Building Block. 2. Taxol CD Ring Unit.

Authors: Uttaro, Jean-Pierre, Audran, Gérard, Monti, Honoré

Source: Journal of Organic Chemistry; April 29 2005, Vol. 70 Issue 9, p3484-3489, 6p

Synthesis and Studies of Potential Inhibitors of CD73 Based on a Triazole Scaffold.

Authors: Grosjean, Félix, Cros‐Perrial, Emeline, Braka, Abdenour, Uttaro, Jean‐Pierre, Chaloin, Laurent, Jordheim, Lars Petter, Peyrottes, Suzanne, Mathé, Christophe

Source: European Journal of Organic Chemistry; 6/7/2022, Vol. 2022 Issue 21, p1-8, 8p

Subject Terms: TRIAZOLES, ENZYME inhibitors, ADENOSINES, ADENOSINE derivatives, TRIAZOLE derivatives

First Enantioselective Synthesis and Absolute Stereochemistry Assignment of New Monocyclic Sesquiterpenes from Artemisia chamaemelifolia.

Authors: Uttaro, Jean-Pierre, Audran, Gérard, Palombo, Elie

Source: Journal of Organic Chemistry; June 27 2003, Vol. 68 Issue 13, p5407-5410, 4p

2‑(Substituted amino)-8-azachromones from 4,6-Diaryl-2-pyridones: A Synthetic Strategy toward Compounds of Broad Structural Diversity.

Authors: Saulnier, Steve¹ (AUTHOR), Ghoteimi, Rayane¹ (AUTHOR), Mathé, Christophe¹ (AUTHOR), Peyrottes, Suzanne¹ (AUTHOR), Uttaro, Jean-Pierre¹ (AUTHOR) jean-pierre.uttaro@umontpellier.fr

Source: Journal of Organic Chemistry. 9/18/2020, Vol. 85 Issue 18, p11778-11793. 16p.

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Synthesis of Substituted 5′‐Aminoadenosine Derivatives and Evaluation of Their Inhibitory Potential toward CD73.

Authors: Ghoteimi, Rayane, Nguyen, >Van Tai, Rahimova, Rahila, Grosjean, Felix, Cros‐Perrial, Emeline, Uttaro, Jean‐Pierre, Mathé, Christophe, Chaloin, Laurent, Jordheim, Lars Petter, Peyrottes, Suzanne

Source: ChemMedChem; 8/6/2019, Vol. 14 Issue 15, p1431-1443, 13p

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Synthesis of {[5-(adenin-9-yl)-2-furyl]methoxy}methyl phosphonic acid and evaluations against human adenylate kinases

Authors: Kaci, Malika, Uttaro, Jean-Pierre, Lefort, Valérie, Mathé, Christophe, El Amri, Chahrazade, Périgaud, Christian

Source: In Bioorganic & Medicinal Chemistry Letters 1 September 2014 24(17):4227-4230

Synthesis and Antiviral Evaluation of 3′‐Fluoro‐4′‐modified‐5′‐norcarbocyclic Nucleoside Phosphonates.

Authors: Geant, Pierre‐Yves, Kaci, Malika, Uttaro, Jean‐Pierre, Périgaud, Christian, Mathé, Christophe

Source: ChemMedChem; 3/5/2019, Vol. 14 Issue 5, p522-526, 5p

Synthesis and Antiviral Evaluation of 3′-Fluoro-5′-norcarbocyclic Nucleoside Phosphonates Bearing Uracil and Cytosine as Potential Antiviral Agents.

Authors: Geant, Pierre-Yves¹ (AUTHOR) pygeant@yahoo.fr, Uttaro, Jean-Pierre¹ (AUTHOR), Périgaud, Christian¹ (AUTHOR), Mathé, Christophe¹ (AUTHOR) christophe.mathe@umontpellier.fr, Seley-Radtke, Katherine (AUTHOR)

Source: Molecules. 8/15/2020, Vol. 25 Issue 16, p3708. 1p. 4 Diagrams.

Subject Terms: *ANTIVIRAL agents, *URACIL derivatives, *PHOSPHONATES, *NUCLEOSIDE derivatives, *URACIL, *CYTOSINE

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Rapid synthesis of carbonucleoside phophonate analogues as potential antiviral agents via a hydrophosphonylation reaction of ethynyl carbocyclic precursors.

Authors: Sidi Mohamed, Bemba, Périgaud, Christian, Peyrottes, Suzanne, Uttaro, Jean-Pierre, Mathé, Christophe

Source: New Journal of Chemistry; 1/15/2018, Vol. 42 Issue 2, p974-979, 6p

Subject Terms: ANTIVIRAL agents, CARBOCYCLIC compounds, CHEMICAL precursors