Replenishing the malaria drug discovery pipeline: Screening and hit evaluation of the MMV Hit Generation Library 1 (HGL1) against asexual blood stage Plasmodium falciparum, using a nano luciferase reporter read-out

Authors: Dechering, Koen J., Timmerman, Martijn, Rensen, Kim, Koolen, Karin M.J., Honarnejad, Saman, Vos, Martijn W., Huijs, Tonnie, Henderson, Rob W.M., Chenu, Elodie, Laleu, Benoît, Montefiore, Bailey C., Segall, Matthew D., Mills, James E.J., Guantai, Eric M., Duffy, James, Duffey, Maëlle

Source: In SLAS Discovery September 2022 27(6):337-348

MAIP: An Open-Source Tool to Enrich High-Throughput Screening Output and Identify Novel, Druglike Molecules with Antimalarial Activity.

Authors: Bosc, Nicolas, Felix, Eloy, Gardner, J. Mark F., Mills, James, Timmerman, Martijn, Asveld, Dennis, Rensen, Kim, Mukherjee, Partha, Das, Rishi, Chenu, Elodie, Besson, Dominique, Burrows, Jeremy N., Duffy, James, Laleu, Benoît, Guantai, Eric M., Leach, Andrew R.

Source: ACS Medicinal Chemistry Letters; 12/14/2023, Vol. 14 Issue 12, p1733-1741, 9p

β-Arrestin-biased signaling of PTH analogs of the type 1 parathyroid hormone receptor

Authors: van der Lee, Miranda M.C., Verkaar, Folkert, Wat, Jesse W.Y., van Offenbeek, Jody, Timmerman, Martijn, Voorneveld, Lonneke, van Lith, Lambertus H.C.J., Zaman, Guido J.R.

Source: In Cellular Signalling February 2013 25(2):527-538

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