Synthesis, in silico modelling, and in vitro biological evaluation of substituted pyrazole derivatives as potential anti-skin cancer, anti-tyrosinase, and antioxidant agents

Authors: Samuel T. Boateng, Tithi Roy, Kara Torrey, Uchechi Owunna, Sergette Banang-Mbeumi, David Basnet, Eleonora Niedda, Alexis D. Alexander, Denzel El Hage, Siriki Atchimnaidu, Bolni Marius Nagalo, Dinesh Aryal, Ann Findley, Navindra P. Seeram, Tatiana Efimova, Mario Sechi, Ronald A. Hill, Hang Ma, Jean Christopher Chamcheu, Siva Murru

Source: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 38, Iss 1 (2023)

Subject Terms: Antitumor agents, apoptosis, tyrosinase inhibition, antioxidant, molecular docking and ADMET, Therapeutics. Pharmacology, RM1-950

File Description: electronic resource

Relation: https://doaj.org/toc/1475-6366; https://doaj.org/toc/1475-6374

Access URL: https://doaj.org/article/6723a7780c15410686963a027f101484

Identification of new fisetin analogs as kinase inhibitors: Data on synthesis and anti-skin cancer activities evaluation

Authors: Tithi Roy, Samuel T. Boateng, Sergette Banang-Mbeumi, Pankaj K. Singh, Pratik Basnet, Roxane-Cherille N. Chamcheu, Federico Ladu, Isabel Chauvin, Vladimir S. Spiegelman, Ronald A. Hill, Konstantin G. Kousoulas, Bolni Marius Nagalo, Anthony L. Walker, Jean Fotie, Siva Murru, Mario Sechi, Jean Christopher Chamcheu

Source: Data in Brief, Vol 35, Iss , Pp 106858- (2021)

Subject Terms: Anticancer evaluation, skin cancers, fisetin analogs, target prediction, computational docking, kinase activities, Computer applications to medicine. Medical informatics, R858-859.7, Science (General), Q1-390

File Description: electronic resource

Relation: http://www.sciencedirect.com/science/article/pii/S2352340921001426; https://doaj.org/toc/2352-3409

Access URL: https://doaj.org/article/8f9eb6ff82c7476a93275e6a6773652e

Intra- and Intermolecular C−S Bond Formation Using a Single Catalytic System: First Direct Access to Arylthiobenzothiazoles.

Authors: Siva Murru¹, Harisadhan Ghosh¹, Santosh K. Sahoo¹, Bhisma K. Patel¹

Source: Organic Letters. Oct2009, Vol. 11 Issue 19, p4254-4257. 4p.

Subject Terms: *COPPER catalysts, *CHEMICAL bonds, *LIGANDS (Chemistry), *ARYLATION, *THIAZOLES, *ORGANIC synthesis

Acyl-isothiocyanates as Efficient Thiocyanate Transfer Reagents.

Authors: Charuta C. Palsuledesai¹, Siva Murru¹, Santosh K. Sahoo¹, Bhisma K. Patel¹

Source: Organic Letters. Aug2009, Vol. 11 Issue 15, p3382-3385. 4p.

Subject Terms: *THIOCYANATES, *CHEMICAL reagents, *BROMIDES, *AMINES, *CHEMICAL reactions, *PROTONS

Self-Assembled Superstructure of Xanthene Derivatives.

Authors: Veerababurao Kavala¹, Siva Murru¹, Bhisma Patel¹, Gopal Das¹

Source: Journal of Chemical Crystallography. Aug2007, Vol. 37 Issue 8, p527-535. 9p.

Subject Terms: *XANTHENE derivatives, *X-ray diffraction, *SOLID state chemistry, *KETONES