Sphingosine 1-phosphate receptor subtype 1 (S1P1) activity in the course of Alzheimer's disease

Authors: Jonatan Martínez-Gardeazabal, Gorka Pereira-Castelo, Marta Moreno-Rodríguez, Alberto Llorente-Ovejero, Manuel Fernández, Iván Fernández-Vega, Iván Manuel, Rafael Rodríguez-Puertas

Source: Neurobiology of Disease, Vol 202, Iss , Pp 106713- (2024)

Subject Terms: S1P1 receptor, Human, Rodents, Brain, [35S]GTPγS, Mapping, Neurosciences. Biological psychiatry. Neuropsychiatry, RC321-571

File Description: electronic resource

Relation: http://www.sciencedirect.com/science/article/pii/S0969996124003152; https://doaj.org/toc/1095-953X

Access URL: https://doaj.org/article/5362973c6a1d4235a640d383951a698b

Synthesis and Evaluation of Serinolamide Derivatives as Sphingosine-1-Phosphate-1 (S1P1) Receptor Agonists

Authors: Sun Jun Park, Jushin Kim, Jaehwan Kim, Yoowon Kim, Elijah Hwejin Lee, Hyeon Jeong Kim, Siwon Kim, Byungeun Kim, Rium Kim, Ji Won Choi, Jong-Hyun Park, Ki Duk Park

Source: Molecules, Vol 27, Iss 9, p 2818 (2022)

Subject Terms: serinolamide A, S1P1 receptor, GPCR, multiple sclerosis, internalization, Organic chemistry, QD241-441

File Description: electronic resource

Relation: https://www.mdpi.com/1420-3049/27/9/2818; https://doaj.org/toc/1420-3049

Access URL: https://doaj.org/article/9513982af7384ce397007a0804d18113

ST-2191, an Anellated Bismorpholino Derivative of Oxy-Fingolimod, Shows Selective S1P1 Agonist and Functional Antagonist Potency In Vitro and In Vivo

Authors: Bisera Stepanovska Tanturovska, Aleksandra Zivkovic, Faik Imeri, Thomas Homann, Burkhard Kleuser, Holger Stark, Andrea Huwiler

Source: Molecules, Vol 26, Iss 17, p 5134 (2021)

Subject Terms: sphingosine 1-phosphate, S1P1 receptor, functional antagonism, lymphopenia, ST-2191, anellated bismorpholino, Organic chemistry, QD241-441

File Description: electronic resource

Relation: https://www.mdpi.com/1420-3049/26/17/5134; https://doaj.org/toc/1420-3049

Access URL: https://doaj.org/article/17a2c0a5ef064ea1b03c5ffcb1344f1f

Effects of multiple-dose ponesimod, a selective S1P1 receptor modulator, on lymphocyte subsets in healthy humans

Authors: Jurcevic S, Juif PE, Hamid C, Greenlaw R, D'Ambrosio D, Dingemanse J

Source: Drug Design, Development and Therapy, Vol Volume11, Pp 123-131 (2016)

Subject Terms: ponesimod, multiple dose, S1P1 receptor, lymphocyte subsets, CD45RA/CCR7, Therapeutics. Pharmacology, RM1-950

File Description: electronic resource

Relation: https://www.dovepress.com/effects-of-multiple-dose-ponesimod-a-selective-s1p1-receptor-modulator-peer-reviewed-article-DDDT; https://doaj.org/toc/1177-8881

Access URL: https://doaj.org/article/759723fb252c43389cb1f1e855f26e74

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