3-Nitroatenolol: First Synthesis, Chiral Resolution and Enantiomers’ Absolute Configuration

Authors: Rosa Sparaco, Pierfrancesco Cinque, Antonia Scognamiglio, Angela Corvino, Giuseppe Caliendo, Ferdinando Fiorino, Elisa Magli, Elisa Perissutti, Vincenzo Santagada, Beatrice Severino, Paolo Luciano, Marcello Casertano, Anna Aiello, Gustavo Yuri Martins Viegas, Gilberto De Nucci, Francesco Frecentese

Source: Molecules, Vol 29, Iss 7, p 1598 (2024)

Subject Terms: 3-nitroatenolol, chiral HPLC, NMR absolute configuration assignment, Riguera’s method, Organic chemistry, QD241-441

File Description: electronic resource

Relation: https://www.mdpi.com/1420-3049/29/7/1598; https://doaj.org/toc/1420-3049

Access URL: https://doaj.org/article/1faca57576ae452e9550a466612b7446

Technological and Physical–Chemical Evaluation of Cotton Gauzes Impregnated with Semisolid Preparations for Wound Healing

Authors: Fabrizio Villapiano, Ritamaria Di Lorenzo, Rosa Sparaco, Elisa Magli, Francesco Frecentese, Sonia Laneri, Alessandra D’Orsi, Valeria Nele, Marco Biondi, Laura Mayol, Virginia Campani, Vincenzo Santagada, Giuseppe De Rosa

Source: Biomedicines, Vol 12, Iss 4, p 777 (2024)

Subject Terms: wound healing, wound dressing, rheology, corneometry, skin energy, Biology (General), QH301-705.5

File Description: electronic resource

Relation: https://www.mdpi.com/2227-9059/12/4/777; https://doaj.org/toc/2227-9059

Access URL: https://doaj.org/article/5e54e6a42b0f47028cbed75bebae7b29

Serotoninergic receptor ligands improve Tamoxifen effectiveness on breast cancer cells

Authors: Maria Rosaria Ambrosio, Elisa Magli, Giuseppe Caliendo, Rosa Sparaco, Paola Massarelli, Vittoria D’Esposito, Teresa Migliaccio, Giusy Mosca, Ferdinando Fiorino, Pietro Formisano

Source: BMC Cancer, Vol 22, Iss 1, Pp 1-14 (2022)

Subject Terms: Serotonin, Breast cancer, Serotoninergic receptor ligands, Tamoxifen resistance, Connective Tissue Growth Factor, Neoplasms. Tumors. Oncology. Including cancer and carcinogens, RC254-282

File Description: electronic resource

Relation: https://doaj.org/toc/1471-2407

Access URL: https://doaj.org/article/1ff550da64d74d238fdea77957c3ed5d

Design, Synthesis and Biological Evaluation of Novel N-Arylpiperazines Containing a 4,5-Dihydrothiazole Ring

Authors: Giorgia Andreozzi, Maria Rosaria Ambrosio, Elisa Magli, Giovanni Maneli, Beatrice Severino, Angela Corvino, Rosa Sparaco, Elisa Perissutti, Francesco Frecentese, Vincenzo Santagada, Anna Leśniak, Magdalena Bujalska-Zadrożny, Giuseppe Caliendo, Pietro Formisano, Ferdinando Fiorino

Source: Pharmaceuticals, Vol 16, Iss 10, p 1483 (2023)

Subject Terms: arylpiperazines, 5-HT1A ligands, binding assays, in vitro assay, cytotoxic activity, Medicine, Pharmacy and materia medica, RS1-441

File Description: electronic resource

Relation: https://www.mdpi.com/1424-8247/16/10/1483; https://doaj.org/toc/1424-8247

Access URL: https://doaj.org/article/f809eadae0904facb28d7ccc4163c291

Synthesis, in vitro and in vivo evaluation of 11C-O-methylated arylpiperazines as potential serotonin 1A (5-HT1A) receptor antagonist radiotracers

Authors: Vidya Narayanaswami, Junchao Tong, Ferdinando Fiorino, Beatrice Severino, Rosa Sparaco, Elisa Magli, Flavia Giordano, Peter M. Bloomfield, Jaya Prabhakaran, J. John Mann, Neil Vasdev, Kenneth Dahl, J. S. Dileep Kumar

Source: EJNMMI Radiopharmacy and Chemistry, Vol 5, Iss 1, Pp 1-17 (2020)

Subject Terms: α1-adrenergic receptor, Carbon-11, 5-HT1A receptor, Serotonin, PET, Medical physics. Medical radiology. Nuclear medicine, R895-920, Therapeutics. Pharmacology, RM1-950

File Description: electronic resource

Relation: http://link.springer.com/article/10.1186/s41181-020-00096-8; https://doaj.org/toc/2365-421X

Access URL: https://doaj.org/article/d04212c45a1c477c855f4b83967b0456

Beneficial Effects of Two Hydrogen Sulfide (H2S)-Releasing Derivatives of Dexamethasone with Antioxidant Activity on Atopic Dermatitis in Mice

Authors: Silvia Abigail Coavoy-Sánchez, Anderson Romério Azevedo Cerqueira, Simone Aparecida Teixeira, Vincenzo Santagada, Giorgia Andreozzi, Angela Corvino, Antonia Scognamiglio, Rosa Sparaco, Giuseppe Caliendo, Beatrice Severino, Soraia Katia Pereira Costa, Luis Carlos Spolidorio, Marcelo Nicolás Muscará

Source: Pharmaceutics, Vol 15, Iss 7, p 1907 (2023)

Subject Terms: hydrogen sulfide, dexamethasone, atopic dermatitis, oxidative stress, Pharmacy and materia medica, RS1-441

File Description: electronic resource

Relation: https://www.mdpi.com/1999-4923/15/7/1907; https://doaj.org/toc/1999-4923

Access URL: https://doaj.org/article/294603bc4e634dcdae188d8f6991cf83

Synthesis, Chiral Resolution and Enantiomers Absolute Configuration of 4-Nitropropranolol and 7-Nitropropranolol

Authors: Rosa Sparaco, Antonia Scognamiglio, Angela Corvino, Giuseppe Caliendo, Ferdinando Fiorino, Elisa Magli, Elisa Perissutti, Vincenzo Santagada, Beatrice Severino, Paolo Luciano, Marcello Casertano, Anna Aiello, Gilberto De Nucci, Francesco Frecentese

Source: Molecules, Vol 28, Iss 1, p 57 (2022)

Subject Terms: 4-nitropropranolol, 7-nitropropranolol, chiral HPLC, NMR absolute configuration assignment, Riguera’s method, Organic chemistry, QD241-441

File Description: electronic resource

Relation: https://www.mdpi.com/1420-3049/28/1/57; https://doaj.org/toc/1420-3049

Access URL: https://doaj.org/article/3ac93dbbe8a24c28ab6152444f9fa139

Synthesis, Docking Studies and Pharmacological Evaluation of Serotoninergic Ligands Containing a 5-Norbornene-2-Carboxamide Nucleus

Authors: Rosa Sparaco, Ewa Kędzierska, Agnieszka A. Kaczor, Anna Bielenica, Elisa Magli, Beatrice Severino, Angela Corvino, Ewa Gibuła-Tarłowska, Jolanta H. Kotlińska, Giorgia Andreozzi, Paolo Luciano, Elisa Perissutti, Francesco Frecentese, Marcello Casertano, Anna Leśniak, Magdalena Bujalska-Zadrożny, Małgorzata Oziębło, Raffaele Capasso, Vincenzo Santagada, Giuseppe Caliendo, Ferdinando Fiorino

Source: Molecules, Vol 27, Iss 19, p 6492 (2022)

Subject Terms: 5-norbornene-2-carboxilic acid, serotonin, arylpiperazine derivatives, 5-HT1A, 5-HT2A and 5-HT2C receptor ligands, Organic chemistry, QD241-441

File Description: electronic resource

Relation: https://www.mdpi.com/1420-3049/27/19/6492; https://doaj.org/toc/1420-3049

Access URL: https://doaj.org/article/7f6a05e3f41942a6b2534e15c918c531

H2S Donors and Their Use in Medicinal Chemistry

Authors: Elisa Magli, Elisa Perissutti, Vincenzo Santagada, Giuseppe Caliendo, Angela Corvino, Gianluca Esposito, Giovanna Esposito, Ferdinando Fiorino, Marco Migliaccio, Antonia Scognamiglio, Beatrice Severino, Rosa Sparaco, Francesco Frecentese

Source: Biomolecules, Vol 11, Iss 12, p 1899 (2021)

Subject Terms: hydrogen sulfide, natural H2S donors, synthetic H2S donors, H2S release, medicinal chemistry, Microbiology, QR1-502

File Description: electronic resource

Relation: https://www.mdpi.com/2218-273X/11/12/1899; https://doaj.org/toc/2218-273X

Access URL: https://doaj.org/article/3f0d2b2493524ef4939b8bf200265b98