[18F]R91150: Improved radiosynthesis and in vivo evaluation as imaging probe for 5-HT2A receptors

Authors: Hoffmann, Chris ^{a, b}, Endepols, Heike ^{a, b, c}, Urusova, Elizaveta A. ^{a, b}, Elchine, Dominik ^a, Neumaier, Felix ^{a, b}, Neumaier, Bernd ^{a, b, ⁎}, Zlatopolskiy, Boris D. ^{a, b}

Source: In European Journal of Medicinal Chemistry 15 March 2025 286

8-Bicycloalkyl-CPFPX derivatives as potent and selective tools for in vivo imaging of the A1 adenosine receptor

Authors: Humpert, Swen, Schneider, Daniela, Bier, Dirk, Schulze, Annette, Neumaier, Felix, Neumaier, Bernd, Holschbach, Marcus

Source: In European Journal of Medicinal Chemistry 5 May 2024 271

Fragmentation of functional resting state brain networks in a transgenic mouse model of tau pathology: A metabolic connectivity study using [18F]FDG-PET

Authors: Endepols, Heike, Anglada-Huguet, Marta, Mandelkow, Eckhard, Neumaier, Bernd, Mandelkow, Eva-Maria, Drzezga, Alexander

Source: In Experimental Neurology February 2024 372

AI-based identification of therapeutic agents targeting GPCRs: introducing ligand type classifiers and systems biologyElectronic supplementary information (ESI) available. See DOI: https://doi.org/10.1039/d3sc02352d

Authors: Goßen, Jonas, Ribeiro, Rui Pedro, Bier, Dirk, Neumaier, Bernd, Carloni, Paolo, Giorgetti, Alejandro, Rossetti, Giulia

Source: Chemical science. 14(32):8651-8661

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100190287739.0x000001&indx=1&recIds=ETOCvdc_100190287739.0x000001

A genetic variation in the adenosine A2A receptor gene contributes to variability in oscillatory alpha power in wake and sleep EEG and A1 adenosine receptor availability in the human brain

Authors: Tichelman, Naemi L., Foerges, Anna L., Elmenhorst, Eva-Maria, Lange, Denise, Hennecke, Eva, Baur, Diego M., Beer, Simone, Kroll, Tina, Neumaier, Bernd, Bauer, Andreas, Landolt, Hans-Peter, Aeschbach, Daniel, Elmenhorst, David

Source: In NeuroImage 15 October 2023 280

Evaluation of the 18F-labeled analog of the therapeutic all-D-enantiomeric peptide RD2 for amyloid β imaging

Authors: Willuweit, Antje, Humpert, Swen, Schöneck, Michael, Endepols, Heike, Burda, Nicole, Gremer, Lothar, Gering, Ian, Kutzsche, Janine, Shah, N.Jon, Langen, Karl-Josef, Neumaier, Bernd, Willbold, Dieter, Drzezga, Alexander

Source: In European Journal of Pharmaceutical Sciences 1 May 2023 184

Transcranial-Direct-Current-Stimulation Accelerates Motor Recovery After Cortical Infarction in Mice: The Interplay of Structural Cellular Responses and Functional Recovery

Authors: Walter, Helene Luise, Pikhovych, Anton, Endepols, Heike, Rotthues, Steffen, Bärmann, Johannes, Backes, Heiko, Hoehn, Mathias, Wiedermann, Dirk, Neumaier, Bernd

Source: Neurorehabilitation and neural repair. 36(10/11):701-714

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCRN630769680&indx=1&recIds=ETOCRN630769680

An ^8^9Zr-Labeled PSMA Tracer for PET/CT Imaging of Prostate Cancer Patients

Authors: Dietlein, Felix, Kobe, Carsten, Vázquez, Sergio Muñoz, Fischer, Thomas, Endepols, Heike, Hohberg, Melanie, Reifegerst, Manuel, Neumaier, Bernd, Schomäcker, Klaus, Drzezga, Alexander E.

Source: Journal of nuclear medicine. 63(4):573-583

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCRN629007694&indx=1&recIds=ETOCRN629007694

MGluR5 and GABAA receptor‐specific parametric PET atlas construction—PET/MR data processing pipeline, validation, and application

Authors: Kaulen, Nicolas, Rajkumar, Ravichandran, Régio Brambilla, Cláudia, Mauler, Jörg, Ramkiran, Shukti, Orth, Linda, Sbaihat, Hasan, Lang, Markus, Wyss, Christine, Rota Kops, Elena, Scheins, Jürgen, Neumaier, Bernd, Ermert, Johannes, Herzog, Hans, Langen, Karl‐Joseph, Lerche, Christoph, Shah, N. Jon, Veselinović, Tanja, Neuner, Irene

Source: Human brain mapping. 43(7):2148-2163

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100146702137.0x000001&indx=1&recIds=ETOCvdc_100146702137.0x000001

Convenient PET-tracer production via SuFEx 18F-fluorination of nanomolar precursor amounts

Authors: Walter, Nils, Bertram, Jan, Drewes, Birte, Bahutski, Victor, Timmer, Marco, Schütz, Markus B., Krämer, Felicia, Neumaier, Felix, Endepols, Heike, Neumaier, Bernd, Zlatopolskiy, Boris D.

Source: In European Journal of Medicinal Chemistry 5 July 2022 237

Do you know your PSMA-tracer? Variability in the biodistribution of different PSMA ligands and its potential impact on defining PSMA-positivity prior to PSMA-targeted therapy.

Authors: Heilinger, Jan, Roth, Katrin Sabine, Weis, Henning, Fink, Antonis, Weindler, Jasmin, Dietlein, Felix, Krapf, Philipp, Schomäcker, Klaus, Neumaier, Bernd, Dietlein, Markus, Drzezga, Alexander, Kobe, Carsten

Source: EJNMMI Research; 1/10/2025, Vol. 15 Issue 1, p1-8, 8p

Subject Terms: PAROTID glands, CANCER relapse, PATIENT selection, LIGANDS (Biochemistry), SPLEEN

Fully Automated Production of (((S)-1-Carboxy-5-(6-([ 18 F]fluoro)-2-methoxynicotinamido)pentyl)carbamoyl)-l-glutamic Acid ([ 18 F]JK-PSMA-7) †.

Authors: Krapf, Philipp, Wicher, Thomas, Zlatopolskiy, Boris D., Ermert, Johannes, Neumaier, Bernd

Source: Pharmaceuticals (14248247); Jan2025, Vol. 18 Issue 1, p119, 14p

Subject Terms: POSITRON emission tomography, RADIOCHEMICAL purification, PROSTATE cancer, RADIOACTIVE tracers, AUTOMATION

Effect of Acute Hypoxia Exposure on the Availability of A1 Adenosine Receptors and Perfusion in the Human Brain.

Authors: Michno, Manuel, Schmitz, Jan, Foerges, Anna L., Beer, Simone, Jordan, Jens, Neumaier, Bernd, Drzezga, Alexander, Aeschbach, Daniel, Bauer, Andreas, Tank, Jens, Weis, Henning, Elmenhorst, Eva-Maria, Elmenhorst, David

Source: Journal of Nuclear Medicine; Jan2025, Vol. 66 Issue 1, p142-149, 8p

Imaging of cerebral tryptophan metabolism using 7-[18F]FTrp-PET in a unilateral Parkinsonian rat model

Authors: Endepols, Heike, Zlatopolskiy, Boris D., Zischler, Johannes, Alavinejad, Nazanin, Apetz, Nadine, Vus, Stefanie, Drzezga, Alexander, Neumaier, Bernd

Source: In NeuroImage 15 February 2022 247

Cerebral A1 adenosine receptor availability in female and male participants and its relationship to sleep

Authors: Pierling, Anna L., Elmenhorst, Eva-Maria, Lange, Denise, Hennecke, Eva, Baur, Diego M., Beer, Simone, Kroll, Tina, Neumaier, Bernd, Aeschbach, Daniel, Bauer, Andreas, Landolt, Hans-Peter, Elmenhorst, David

Source: In NeuroImage 15 December 2021 245

Production cross-section measurements of proton-induced reactions on natural tantalum in the 0.3 GeV–1.7 GeV energy range

Authors: Duchemin, Charlotte, Cocolios, Thomas E., Dockx, Kristof, Farooq-Smith, Gregory J., Felden, Olaf, Formento-Cavaier, Roberto, Gebel, Ralf, Köster, Ulli, Neumaier, Bernd, Scholten, Bernhard, Spahn, Ingo, Spellerberg, Stefan, Stamati, Maria E., Stegemann, Simon, Verhoeven, Hannelore

Source: In Applied Radiation and Isotopes December 2021 178

Design, synthesis and biological evaluation of Tozadenant analogues as adenosine A2A receptor ligands

Authors: Renk, Dana R., Skraban, Marcel, Bier, Dirk, Schulze, Annette, Wabbals, Erika, Wedekind, Franziska, Neumaier, Felix, Neumaier, Bernd, Holschbach, Marcus

Source: In European Journal of Medicinal Chemistry 15 March 2021 214

Radiosynthesis and evaluation of 18F-labeled dopamine D4-receptor ligands

Authors: Willmann, Michael, Ermert, Johannes, Prante, Olaf, Hübner, Harald, Gmeiner, Peter, Neumaier, Bernd

Source: In Nuclear Medicine and Biology January 2021 92:43-52

18F-Labeled magnetic nanovectors for bimodal cellular imagingElectronic supplementary information (ESI) available. See DOI: 10.1039/d1bm00616a

Authors: Schütz, Markus B., Renner, Alexander M., Ilyas, Shaista, Lê, Khan, Guliyev, Mehrab, Krapf, Philipp, Neumaier, Bernd, Mathur, Sanjay

Source: Biomaterials science. 9(13):4717-4727

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100122055884.0x000001&indx=1&recIds=ETOCvdc_100122055884.0x000001

One-Stop Shop: ^1^8F-Flortaucipir PET Differentiates Amyloid-Positive and -Negative Forms of Neurodegenerative Diseases

Authors: Hammes, Jochen, Bischof, Gérard N., Bohn, Karl P., Onur, Özgür, Schneider, Anja, Fliessbach, Klaus, Hönig, Merle C, Jessen, Frank, Neumaier, Bernd, Drzezga, Alexander

Source: Journal of nuclear medicine. 62(2):240-246

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCRN625675168&indx=1&recIds=ETOCRN625675168