Numb-associated kinases are required for SARS-CoV-2 infection and are cellular targets for antiviral strategies

Authors: Karim, Marwah, Saul, Sirle, Ghita, Luca, Sahoo, Malaya Kumar, Ye, Chengjin, Bhalla, Nishank, Lo, Chieh-Wen, Jin, Jing, Park, Jun-Gyu, Martinez-Gualda, Belén, East, Michael Patrick, Johnson, Gary L., Pinsky, Benjamin A., Martinez-Sobrido, Luis, Asquith, Christopher R.M., Narayanan, Aarthi, De Jonghe, Steven, Einav, Shirit

Source: In Antiviral Research August 2022 204

Organotropic dendrons with high potency as HIV-1, HIV-2 and EV-A71 cell entry inhibitors

Authors: Martí-Marí, Olaia, Martínez-Gualda, Belén, Fernández-Barahona, Irene, Mills, Alberto, Abdelnabi, Rana, Noppen, Sam, Neyts, Johan, Schols, Dominique, Camarasa, María-José, Herranz, Fernando, Gago, Federico, San-Félix, Ana

Source: In European Journal of Medicinal Chemistry 5 July 2022 237

Discovery of 3-phenyl- and 3-N-piperidinyl-isothiazolo[4,3-b]pyridines as highly potent inhibitors of cyclin G-associated kinase

Authors: Martinez-Gualda, Belén, Saul, Sirle, Froeyen, Mathy, Schols, Dominique, Herdewijn, Piet, Einav, Shirit, De Jonghe, Steven

Source: In European Journal of Medicinal Chemistry 5 March 2021 213

A patent review of adaptor associated kinase 1 (AAK1) inhibitors (2013-present)

Authors: Martinez-Gualda, Belén, Schols, Dominique, De Jonghe, Steven

Source: Expert opinion on therapeutic patents. 31(10):911-936

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100130175593.0x000001&indx=1&recIds=ETOCvdc_100130175593.0x000001

Structure-activity relationship study of the pyridine moiety of isothiazolo[4,3-b]pyridines as antiviral agents targeting cyclin G-associated kinase

Authors: Martinez-Gualda, Belén, Pu, Szu-Yuan, Froeyen, Mathy, Herdewijn, Piet, Einav, Shirit, De Jonghe, Steven

Source: In Bioorganic & Medicinal Chemistry 1 January 2020 28(1)

Structure-activity relationship studies on a Trp dendrimer with dual activities against HIV and enterovirus A71. Modifications on the amino acid

Authors: Martínez-Gualda, Belén, Sun, Liang, Rivero-Buceta, Eva, Flores, Aida, Quesada, Ernesto, Balzarini, Jan, Noppen, Sam, Liekens, Sandra, Schols, Dominique, Neyts, Johan, Leyssen, Pieter, Mirabelli, Carmen, Camarasa, María-José, San-Félix, Ana

Source: In Antiviral Research March 2017 139:32-40

Discovery of 3-phenyl- and 3-N-piperidinyl-isothiazolo[4, 3-b]pyridines as highly potent inhibitors of cyclin G-associated kinase

Authors: Martinez-Gualda, Belén, Saul, Sirle, Froeyen, Mathy, Schols, Dominique, Herdewijn, Piet, Einav, Shirit, De Jonghe, Steven

Source: European journal of medicinal chemistry. 213

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100136562006.0x000001&indx=1&recIds=ETOCvdc_100136562006.0x000001

Structure-activity relationship study of the pyridine moiety of isothiazolo[4, 3-b]pyridines as antiviral agents targeting cyclin G-associated kinase

Authors: Martinez-Gualda, Belén, Pu, Szu-Yuan, Froeyen, Mathy, Herdewijn, Piet, Einav, Shirit, De Jonghe, Steven

Source: Bioorganic & medicinal chemistry. 28(1)

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100098455862.0x000001&indx=1&recIds=ETOCvdc_100098455862.0x000001

Modifications in the branched arms of a class of dual inhibitors of HIV and EV71 replication expand their antiviral spectrum

Authors: Martínez-Gualda, Belén, Sun, Liang, Martí-Marí, Olaia, Mirabelli, Carmen, Delang, Leen, Neyts, Johan, Schols, Dominique, Camarasa, María-José, San-Félix, Ana

Source: In Antiviral Research August 2019 168:210-214

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