Benchmarking Australian Enabling Programs for a National Framework of Standards. A Practice Report

Authors: Davis, Charmaine (ORCID 0000-0003-2194-2307), Cook, Chris (ORCID 0000-0001-9339-638X), Syme, Suzi (ORCID 0000-0001-8633-0286), Dempster, Sarah, Duffy, Lisa (ORCID 0000-0002-8681-9206), Hattam, Sarah (ORCID 0000-0002-3667-6753), Lambrinidis, George (ORCID 0000-0001-8771-1304), Lawson, Kathy, Levy, Stuart (ORCID 0000-0002-8845-8870)

Source: Student Success. 2023 14(2):41-49.

Peer Reviewed: Y

Page Count: 9

Descriptors: Benchmarking, National Standards, Alignment (Education), Universities, Institutional Cooperation, Foreign Countries, Access to Education, Guidelines, Educational Practices

Geographic Terms: Australia

Accurate calculation of affinity changes to the close state of influenza A M2 transmembrane domain in response to subtle structural changes of adamantyl amines using free energy perturbation methods in different lipid bilayers

Authors: Georgiou, Kyriakos ^a, Konstantinidi, Athina ^a, Hutterer, Johanna ^b, Freudenberger, Kathrin ^b, Kolarov, Felix ^{b, c}, Lambrinidis, George ^a, Stylianakis, Ioannis ^a, Stampelou, Margarita ^a, Gauglitz, Günter ^b, Kolocouris, Antonios ^{a, ⁎}

Source: In BBA - Biomembranes February 2024 1866(2)

Uracil/H+ Symport by FurE Refines Aspects of the Rocking-bundle Mechanism of APC-type Transporters

Authors: Zantza, Iliana, Pyrris, Yiannis, Raniolo, Stefano, Papadaki, Georgia F., Lambrinidis, George, Limongelli, Vittorio, Diallinas, George, Mikros, Emmanuel

Source: In Journal of Molecular Biology 1 October 2023 435(19)

Investigation of Tumor Cells and Receptor-Ligand Simulation Models for the Development of PET Imaging Probes Targeting PSMA and GRPR and a Possible Crosstalk between the Two Receptors

Authors: Liolios, Christos, Patsis, Christos, Lambrinidis, George, Tzortzini, Efpraxia, Roscher, Mareike, Bauder-Wüst, Ulrike, Kolocouris, Antonios, Kopka, Klaus

Source: Molecular pharmaceutics. 19(7):2231-2247

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCRN629737933&indx=1&recIds=ETOCRN629737933

Towards New Scaffolds for Antimicrobial Activity—In Silico/In Vitro Workflow Introducing New Lead Compounds.

Authors: Mangana, Maria, Lambrinidis, George, Kostakis, Ioannis K., Kalpaktsi, Ioanna, Sagnou, Marina, Nicolaou, Chrysoula, Mikros, Emmanuel, Chatzipanagiotou, Stylianos, Ioannidis, Anastasios

Source: Antibiotics (2079-6382); Jan2025, Vol. 14 Issue 1, p11, 11p

Subject Terms: DRUG discovery, CHEMICAL libraries, DRUG resistance in bacteria, DRUG design, GRAM-negative bacteria

Design, synthesis, and biological evaluation of new raloxifene analogues of improved antagonist activity and endometrial safety

Authors: Lambrinidis, George, Gouedard, Cedric, Stasinopoulou, Sotiria, Angelopoulou, Angeliki, Ganou, Vassiliki, Meligova, Aggeliki K., Mitsiou, Dimitra J., Marakos, Panagiotis, Pouli, Nicole, Mikros, Emmanuel, Alexis, Michael N.

Source: In Bioorganic Chemistry January 2021 106

Multi-objective optimization methods in novel drug design

Authors: Lambrinidis, George, Tsantili-Kakoulidou, Anna

Source: Expert opinion on drug discovery. 16(6):647-658

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100121402022.0x000001&indx=1&recIds=ETOCvdc_100121402022.0x000001

Novel Carbamοyloxy Analogues of Tamoxifen: Synthesis, Molecular Docking and Bioactivity Evaluation

Authors: Kasiotis, Konstantinos M., Lambrinidis, George, Fokialakis, Nikolas, Haroutounian, Serkos A.

Source: Letters in drug design & discovery. 18(5):422-428

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100129242631.0x000001&indx=1&recIds=ETOCvdc_100129242631.0x000001

Synthesis and Preclinical Evaluation of a Bispecific PSMA-617/RM2 Heterodimer Targeting Prostate Cancer.

Authors: Liolios, Christos, Bouziotis, Danai, Sihver, Wiebke, Schäfer, Martin, Lambrinidis, George, Salvanou, Evangelia-Alexandra, Bauder-Wüst, Ulrike, Benesova, Martina, Kopka, Klaus, Kolocouris, Antonios, Bouziotis, Penelope

Source: ACS Medicinal Chemistry Letters; 11/14/2024, Vol. 15 Issue 11, p1970-1978, 9p

Steroid sulfatase inhibiting lanostane triterpenes – Structure activity relationship and in silico insights

Authors: Grienke, Ulrike, Kaserer, Teresa, Kirchweger, Benjamin, Lambrinidis, George, Kandel, Ralph T., Foster, Paul A., Schuster, Daniela, Mikros, Emmanuel, Rollinger, Judith M.

Source: In Bioorganic Chemistry January 2020 95

Cytosolic N- and C-Termini of the Aspergillus nidulans FurE Transporter Contain Distinct Elements that Regulate by Long-Range Effects Function and Specificity

Authors: Papadaki, Georgia F., Lambrinidis, George, Zamanos, Andreas, Mikros, Emmanuel, Diallinas, George

Source: In Journal of Molecular Biology 6 September 2019 431(19):3827-3844

Adiponectin Signaling and Impaired GTPase Rab5 Expression in Adipocytes of Adolescents with Obesity

Authors: Karvela, Alexia, Kostopoulou, Eirini, Rojas Gil, Andrea Paola, Avgeri, Aikaterini, Pappa, Aliki, Barrios, Vicente, Lambrinidis, George, Dimopoulos, Ioannis, Georgiou, George, Argente, Jesús, Spiliotis, Bessie

Source: Hormone research in pædiatrics. 93(5):287-296

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100111106621.0x000001&indx=1&recIds=ETOCvdc_100111106621.0x000001

X-ray Crystal Structures of the Influenza M2 Proton Channel Drug-Resistant V27A Mutant Bound to a Spiro-Adamantyl Amine Inhibitor Reveal the Mechanism of Adamantane Resistance

Authors: Thomaston, Jessica L., Konstantinidi, Athina, Liu, Lijun, Lambrinidis, George, Tan, Jingquan, Caffrey, Martin, Wang, Jun, Degrado, William F., Kolocouris, Antonios

Source: Biochemistry. 59(4):628-634

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCRN623188691&indx=1&recIds=ETOCRN623188691

Hit-to-Lead Optimization of Heterocyclic Carbonyloxycarboximidamides as Selective Antagonists at Human Adenosine A3 Receptor.

Authors: Huang, Xianglin, Chorianopoulou, Anna, Kalkounou, Panagoula, Georgiou, Maria, Pousias, Athanasios, Davies, Amy, Pearce, Abigail, Harris, Matthew, Lambrinidis, George, Marakos, Panagiotis, Pouli, Nicole, Kolocouris, Antonios, Lougiakis, Nikolaos, Ladds, Graham

Source: Journal of Medicinal Chemistry; 8/8/2024, Vol. 67 Issue 15, p13117-13146, 30p

The olive constituent oleuropein, as a PPARα agonist, markedly reduces serum triglycerides

Authors: Malliou, Foteini, Andreadou, Ioanna, Gonzalez, Frank J., Lazou, Antigone, Xepapadaki, Eva, Vallianou, Ioanna, Lambrinidis, George, Mikros, Emmanuel, Marselos, Marios, Skaltsounis, Alexios-Leandros, Konstandi, Maria

Source: In The Journal of Nutritional Biochemistry September 2018 59:17-28

Structure-activity relationships in fungal nucleobases transporters as dissected by the inhibitory effects of novel purine analogues

Authors: Gavriil, Efthymios-Spyridon, Dimitrakis, Spyridon, Papadaki, Georgia, Balaska, Sophia, Lambrinidis, George, Lougiakis, Nikolaos, Marakos, Panagiotis, Diallinas, George, Pouli, Nicole, Mikros, Emmanuel

Source: In European Journal of Medicinal Chemistry 5 August 2018 156:240-251

Discovery of Novel Adenosine Receptor Antagonists through a Combined Structure- and Ligand-Based Approach Followed by Molecular Dynamics Investigation of Ligand Binding Mode

Authors: Lagarias, Panagiotis, Vrontaki, Eleni, Lambrinidis, George, Stamatis, Dimitrios, Convertino, Marino, Ortore, Gabriella, Mavromoustakos, Thomas, Klotz, Karl-Norbert, Kolocouris, Antonios

Source: JOURNAL OF CHEMICAL INFORMATION AND MODELING. 58(4):794-815

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCRN632678073&indx=1&recIds=ETOCRN632678073

In Silico Screening of Compound Libraries Using a Consensus of Orthogonal Methodologies

Authors: Myrianthopoulos, Vassilios, Lambrinidis, George, Mikros, Emmanuel

Source: Methods in molecular biology. 1824:261-278

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCRN616802584&indx=1&recIds=ETOCRN616802584

Challenges with multi-objective QSAR in drug discovery

Authors: Lambrinidis, George, Tsantili-Kakoulidou, Anna

Source: Expert opinion on drug discovery. 13(9):851-859

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100102910541.0x000001&indx=1&recIds=ETOCvdc_100102910541.0x000001

Design and synthesis of purine analogues as highly specific ligands for FcyB, a ubiquitous fungal nucleobase transporter

Authors: Lougiakis, Nikolaos, Gavriil, Efthymios-Spyridon, Kairis, Markelos, Sioupouli, Georgia, Lambrinidis, George, Benaki, Dimitra, Krypotou, Emilia, Mikros, Emmanuel, Marakos, Panagiotis, Pouli, Nicole, Diallinas, George

Source: In Bioorganic & Medicinal Chemistry 15 November 2016 24(22):5941-5952