Pharmacological characterization of 3, 4-methylenedioxyamphetamine (MDA) analogs and two amphetamine-based compounds: N, α-DEPEA and DPIA

Authors: Kolaczynska, Karolina E., Ducret, Paula, Trachsel, Daniel, Hoener, Marius C., Liechti, Matthias E., Luethi, Dino

Source: European neuropsychopharmacology. 59:9-22

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100164928998.0x000001&indx=1&recIds=ETOCvdc_100164928998.0x000001

Trace amine-associated receptors (TAARs)2-9 knockout mice exhibit reduced wakefulness and disrupted REM sleep.

Authors: Park, Sunmee, Heu, Jasmine, Scheldrup, Gavin, Tisdale, Ryan K., Sun, Yu, Haire, Meghan, Ma, Shun-Chieh, Hoener, Marius C., Kilduff, Thomas S.

Source: Frontiers in Psychiatry; 2025, p1-14, 14p

Subject Terms: SLEEP, RAPID eye movement sleep, SLEEP deprivation, TYROSINE hydroxylase, KNOCKOUT mice

Pharmacological characterization of 3,4-methylenedioxyamphetamine (MDA) analogs and two amphetamine-based compounds: N,α-DEPEA and DPIA

Authors: Kolaczynska, Karolina E., Ducret, Paula, Trachsel, Daniel, Hoener, Marius C., Liechti, Matthias E., Luethi, Dino

Source: In European Neuropsychopharmacology June 2022 59:9-22

Effect of the TAAR1 Partial Agonist Ralmitaront on Presynaptic Dopamine Synthesis Capacity Measured Using [ 18 F]DOPA PET in Naïve and Cocaine-Treated Mice.

Authors: Bonsall, David R., Kokkinou, Michelle, Halff, Els F., Rutigliano, Grazia, Tang, Sac-Pham, Veronese, Mattia, Irvine, Elaine E., Withers, Dominic J., Wells, Lisa A., Natesan, Sridhar, Gerlach, Irene, Holiga, Štefan, Hoener, Marius C., Howes, Oliver D.

Source: Molecular Imaging; 12/18/2024, Vol. 23, p1-5, 5p

Subject Terms: DOPAMINE agonists, POSITRON emission tomography, CAPACITY (Law), DOPA, COCAINE, DOPAMINE

Wakefulness Induced by TAAR1 Partial Agonism in Mice Is Mediated Through Dopaminergic Neurotransmission †.

Authors: Park, Sunmee, Heu, Jasmine, Hoener, Marius C., Kilduff, Thomas S.

Source: International Journal of Molecular Sciences; Nov2024, Vol. 25 Issue 21, p11351, 15p

Subject Terms: SLEEP latency, RAPID eye movement sleep, NEURAL transmission, SLEEP, WAKEFULNESS, ELECTROENCEPHALOGRAPHY, NON-REM sleep

Pharmacological profiles of compounds in preworkout supplements (“boosters”)

Authors: Rickli, Anna, Hoener, Marius C., Liechti, Matthias E.

Source: In European Journal of Pharmacology 15 September 2019 859

Monoamine receptor interaction profiles of 4-aryl-substituted 2,5-dimethoxyphenethylamines (2C-BI derivatives)

Authors: Luethi, Dino, Widmer, Robert, Trachsel, Daniel, Hoener, Marius C., Liechti, Matthias E.

Source: In European Journal of Pharmacology 15 July 2019 855:103-111

Cytochrome P450 enzymes contribute to the metabolism of LSD to nor-LSD and 2-oxo-3-hydroxy-LSD: Implications for clinical LSD use

Authors: Luethi, Dino, Hoener, Marius C., Krähenbühl, Stephan, Liechti, Matthias E., Duthaler, Urs

Source: In Biochemical Pharmacology June 2019 164:129-138

Pharmacological characterization of the aminorex analogs 4-MAR, 4,4′-DMAR, and 3,4-DMAR

Authors: Rickli, Anna, Kolaczynska, Karolina, Hoener, Marius C., Liechti, Matthias E.

Source: In Neurotoxicology May 2019 72:95-100

Electrophysiological Phenotype in Angelman Syndrome Differs Between Genotypes

Authors: Frohlich, Joel, Miller, Meghan T., Bird, Lynne M., Garces, Pilar, Purtell, Hannah, Hoener, Marius C., Philpot, Benjamin D., Sidorov, Michael S., Tan, Wen-Hann, Hernandez, Maria-Clemencia, Rotenberg, Alexander, Jeste, Shafali S., Krishnan, Michelle, Khwaja, Omar, Hipp, Joerg F.

Source: In Biological Psychiatry 1 May 2019 85(9):752-759

Stereochemistry of phase-1 metabolites of mephedrone determines their effectiveness as releasers at the serotonin transporter

Authors: Mayer, Felix P., Cintulova, Daniela, Pittrich, Dorothea A., Wimmer, Laurin, Luethi, Dino, Holy, Marion, Jaentsch, Kathrin, Tischberger, Sonja, Gmeiner, Guenter, Hoener, Marius C., Liechti, Matthias E., Mihovilovic, Marko D., Sitte, Harald H.

Source: In Neuropharmacology April 2019 148:199-209

Activation of trace amine-associated receptor 1 attenuates schedule-induced polydipsia in rats

Authors: Sukhanov, Ilya, Dorotenko, Artem, Dolgorukova, Antonina, Hoener, Marius C., Gainetdinov, Raul R., Bespalov, Anton Yu.

Source: In Neuropharmacology January 2019 144:184-192

The psychostimulant (±)-cis-4,4′-dimethylaminorex (4,4′-DMAR) interacts with human plasmalemmal and vesicular monoamine transporters

Authors: Maier, Julian, Mayer, Felix P., Luethi, Dino, Holy, Marion, Jäntsch, Kathrin, Reither, Harald, Hirtler, Lena, Hoener, Marius C., Liechti, Matthias E., Pifl, Christian, Brandt, Simon D., Sitte, Harald H.

Source: In Neuropharmacology August 2018 138:282-291

Trace Amines and Their Receptors

Authors: Gainetdinov, Raul R. ^*, Hoener, Marius C., Berry, Mark D.

Source: In Pharmacological Reviews July 2018 70(3):549-620

Monoamine receptor interaction profiles of 4-thio-substituted phenethylamines (2C-T drugs)

Authors: Luethi, Dino, Trachsel, Daniel, Hoener, Marius C., Liechti, Matthias E.

Source: In Neuropharmacology 15 May 2018 134 Part A:141-148

Pharmacological profile of methylphenidate-based designer drugs

Authors: Luethi, Dino, Kaeser, Philine J., Brandt, Simon D., Krähenbühl, Stephan, Hoener, Marius C., Liechti, Matthias E.

Source: In Neuropharmacology 15 May 2018 134 Part A:133-140

Pharmacological profile of mephedrone analogs and related new psychoactive substances

Authors: Luethi, Dino, Kolaczynska, Karolina E., Docci, Luca, Krähenbühl, Stephan, Hoener, Marius C., Liechti, Matthias E.

Source: In Neuropharmacology 15 May 2018 134 Part A:4-12

Effects of the new psychoactive substances diclofensine, diphenidine, and methoxphenidine on monoaminergic systems

Authors: Luethi, Dino, Hoener, Marius C., Liechti, Matthias E.

Source: In European Journal of Pharmacology 15 January 2018 819:242-247

TAAR1 levels and sub-cellular distribution are cell line but not breast cancer subtype specific

Authors: Pitts, Mallory S., McShane, Josh N., Hoener, Marius C., Christian, Sherri L., Berry, Mark D.

Source: Histochemistry and cell biology. 152(2):155-166

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100141510531.0x000001&indx=1&recIds=ETOCvdc_100141510531.0x000001

Monoamine receptor interaction profiles of 4-aryl-substituted 2, 5-dimethoxyphenethylamines (2C-BI derivatives)

Authors: Luethi, Dino, Widmer, Robert, Trachsel, Daniel, Hoener, Marius C., Liechti, Matthias E.

Source: European journal of pharmacology. 855:103-111

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100081999680.0x000001&indx=1&recIds=ETOCvdc_100081999680.0x000001