Design and synthesis of 4-amino-2′,4′-dihydroxyindanone derivatives as potent inhibitors of tyrosinase and melanin biosynthesis in human melanoma cells

Authors: Lazinski, Leticia M., Beaumet, Morane, Roulier, Brayan, Gay, Rémy, Royal, Guy, Maresca, Marc, Haudecoeur, Romain

Source: In European Journal of Medicinal Chemistry 15 February 2024 266

Aurones and derivatives as promising New Delhi metallo-β-lactamase (NDM-1) inhibitors

Authors: Caburet, Jérémy, Verdirosa, Federica, Moretti, Matis, Roulier, Brayan, Simoncelli, Giorgia, Haudecoeur, Romain, Ghazi, Somayeh, Jamet, Hélène, Docquier, Jean-Denis, Boucherle, Benjamin, Peuchmaur, Marine

Source: In Bioorganic & Medicinal Chemistry 1 January 2024 97

Catechol-mimicking transition-state analogues as non-oxidizable inhibitors of tyrosinases

Authors: Beaumet, Morane, Lazinski, Leticia M., Maresca, Marc, Haudecoeur, Romain

Source: In European Journal of Medicinal Chemistry 5 November 2023 259

Tyrosinase Inhibition and Antimelanogenic Effects of Resorcinol‐Containing Compounds.

Authors: Beaumet, Morane, Lazinski, Leticia M., Maresca, Marc, Haudecoeur, Romain

Source: ChemMedChem; 12/2/2024, Vol. 19 Issue 23, p1-18, 18p

Targeting different binding sites in the CFTR structures allows to synergistically potentiate channel activity

Authors: Froux, Lionel, Elbahnsi, Ahmad, Boucherle, Benjamin, Billet, Arnaud, Baatallah, Nesrine, Hoffmann, Brice, Alliot, Julien, Zelli, Renaud, Zeinyeh, Wael, Haudecoeur, Romain, Chevalier, Benoit, Fortuné, Antoine, Mirval, Sandra, Simard, Christophe, Lehn, Pierre, Mornon, Jean-Paul, Hinzpeter, Alexandre, Becq, Frédéric, Callebaut, Isabelle, Décout, Jean-Luc

Source: In European Journal of Medicinal Chemistry 15 March 2020 190

Resorcinol-based hemiindigoid derivatives as human tyrosinase inhibitors and melanogenesis suppressors in human melanoma cells

Authors: Roulier, Brayan, Rush, Inbal, Lazinski, Leticia M., Pérès, Basile, Olleik, Hamza, Royal, Guy, Fishman, Ayelet, Maresca, Marc, Haudecoeur, Romain

Source: European journal of medicinal chemistry. 246

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100178231494.0x000001&indx=1&recIds=ETOCvdc_100178231494.0x000001

Aurone derivatives as promising antibacterial agents against resistant Gram-positive pathogens

Authors: Olleik, Hamza, Yahiaoui, Samir, Roulier, Brayan, Courvoisier-Dezord, Elise, Perrier, Josette, Pérès, Basile, Hijazi, Akram, Baydoun, Elias, Raymond, Josette, Boumendjel, Ahcène, Maresca, Marc, Haudecoeur, Romain

Source: In European Journal of Medicinal Chemistry 1 March 2019 165:133-141

Piperidinyl-embeded chalcones possessing anti PI3Kδ inhibitory properties exhibit anti-atopic properties in preclinical models

Authors: Dumontet, Charles, Beck, Guillaume, Gardebien, Fabrice, Haudecoeur, Romain, Mathé, Doriane, Matera, Eva-Laure, Tourette, Anne, Mattei, Eve, Esmenjaud, Justine, Boyère, Cédric, Nurisso, Alessandra, Peuchmaur, Marine, Pérès, Basile, Bouchaud, Grégory, Magnan, Antoine, Monneret, Guillaume, Boumendjel, Ahcène

Source: In European Journal of Medicinal Chemistry 5 October 2018 158:405-413

Occurrences, biosynthesis and properties of aurones as high-end evolutionary products

Authors: Boucherle, Benjamin, Peuchmaur, Marine, Boumendjel, Ahcène, Haudecoeur, Romain

Source: In Phytochemistry October 2017 142:92-111

Expanding Chemical Frontiers: Approaches for Generating Diverse and Bioactive Natural Product‐Like Compounds Libraries from Extracts.

Authors: Beato, Aurélien¹ (AUTHOR), Haudecoeur, Romain¹ (AUTHOR), Boucherle, Benjamin¹ (AUTHOR), Peuchmaur, Marine¹ (AUTHOR) marine.peuchmaur@univ-grenoble-alpes.fr

Source: Chemistry - A European Journal. 5/8/2024, Vol. 30 Issue 26, p1-20. 20p.

Subject Terms: *CHEMICAL libraries, *SYNTHETIC products, *NATURAL products, *CHEMICAL engineering, *CHEMICAL engineers, *NITROGEN

Traditional uses, phytochemistry and pharmacological properties of African Nauclea species: A review

Authors: Haudecoeur, Romain, Peuchmaur, Marine, Pérès, Basile, Rome, Maxime, Taïwe, Germain Sotoing, Boumendjel, Ahcène, Boucherle, Benjamin

Source: Journal of ethnopharmacology. 212:106-136

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100131031812.0x000001&indx=1&recIds=ETOCvdc_100131031812.0x000001

Glycosyl‐Substituted Dicarboxylates as Detergents for the Extraction, Overstabilization, and Crystallization of Membrane Proteins

Authors: Nguyen, Kim‐Anh, Peuchmaur, Marine, Magnard, Sandrine, Haudecoeur, Romain, Boyère, Cédric, Mounien, Saravanan, Benammar, Ikram, Zampieri, Veronica, Igonet, Sébastien, Chaptal, Vincent, Jawhari, Anass, Boumendjel, Ahcène, Falson, Pierre

Source: Angewandte Chemie international edition. 57(11):2948-2952

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100083950688.0x000001&indx=1&recIds=ETOCvdc_100083950688.0x000001

Design and Synthesis of Novel Amino and Acetamidoaurones with Antimicrobial Activities.

Authors: Di Maio, Attilio, Olleik, Hamza, Courvoisier-Dezord, Elise, Guillier, Sophie, Neulat-Ripoll, Fabienne, Haudecoeur, Romain, Bolla, Jean-Michel, Casanova, Magali, Cavalier, Jean-François, Canaan, Stéphane, Pique, Valérie, Charmasson, Yolande, Baydoun, Elias, Hijazi, Akram, Perrier, Josette, Maresca, Marc, Robin, Maxime

Source: Antibiotics (2079-6382); Apr2024, Vol. 13 Issue 4, p300, 19p

Subject Terms: ANTI-infective agents, CYTOTOXINS, AMINO group, AURONES, ANTIBACTERIAL agents, PEPTIDE antibiotics

B-ring modified aurones as promising allosteric inhibitors of hepatitis C virus RNA-dependent RNA polymerase

Authors: Meguellati, Amel, Ahmed-Belkacem, Abdelhakim, Yi, Wei, Haudecoeur, Romain, Crouillère, Marie, Brillet, Rozenn, Pawlotsky, Jean-Michel, Boumendjel, Ahcène, Peuchmaur, Marine

Source: In European Journal of Medicinal Chemistry 10 June 2014 80:579-592

Recombinant Tyrosinase from Polyporus arcularius: Overproduction in Escherichia coli, Characterization, Use in a Study of Aurones as Tyrosinase Effectors

Authors: Marková, Eva, Kotik, Michael, Křenková, Alena, Man, Petr, Haudecoeur, Romain, Boumendjel, Ahcène, Hardré, Renaud, Mekmouche, Yasmina, Courvoisier-Dezord, Elise, Réglier, Marius

Source: Journal of agricultural and food chemistry. 64(14):2925-2931

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCRN605855245&indx=1&recIds=ETOCRN605855245

Refinement of arylthiosemicarbazone pharmacophore in inhibition of mushroom tyrosinase

Authors: Yi, Wei, Dubois, Carole, Yahiaoui, Samir, Haudecoeur, Romain, Belle, Catherine, Song, Huacan, Hardré, Renaud, Réglier, Marius, Boumendjel, Ahcène

Source: In European Journal of Medicinal Chemistry 2011 46(9):4330-4335

Bioactive Aurones, Indanones, and Other Hemiindigoid Scaffolds: Medicinal Chemistry and Photopharmacology Perspectives.

Authors: Lazinski, Leticia M., Royal, Guy, Robin, Maxime, Maresca, Marc, Haudecoeur, Romain

Source: Journal of Medicinal Chemistry; 10/13/2022, Vol. 65 Issue 19, p12594-12625, 32p

β‑Carboline as a Privileged Scaffold for Multitarget Strategies in Alzheimer's Disease Therapy.

Authors: Beato, Aurélien, Gori, Anthonin, Boucherle, Benjamin, Peuchmaur, Marine, Haudecoeur, Romain

Source: Journal of Medicinal Chemistry; 2/11/2021, Vol. 64 Issue 3, p1392-1422, 31p

Advances in the Design of Genuine Human Tyrosinase Inhibitors for Targeting Melanogenesis and Related Pigmentations.

Authors: Roulier, Brayan, Pérès, Basile, Haudecoeur, Romain

Source: Journal of Medicinal Chemistry; 11/25/2020, Vol. 63 Issue 22, p13428-13443, 16p

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