Scaffold modifications to the 4-(4,4-dimethylpiperidinyl) 2,6-dimethylpyridinyl class of HIV-1 allosteric integrase inhibitors

Authors: Parcella, Kyle, Patel, Manoj, Tu, Yong, Eastman, Kyle, Peese, Kevin, Gillis, Eric, Belema, Makonen, Dicker, Ira B., McAuliffe, Brian, Ding, Bo, Falk, Paul, Simmermacher, Jean, Parker, Dawn D., Sivaprakasam, Prasanna, Khan, Javed A., Kish, Kevin, Lewis, Hal, Hanumegowda, Umesh, Jenkins, Susan, Kadow, John F., Krystal, Mark, Meanwell, Nicholas A., Naidu, B. Narasimhulu

Source: In Bioorganic & Medicinal Chemistry 1 August 2022 67

Racial and ethnic disparities in H1N1 vaccine uptake in Medicaid: Lessons learned for a COVID-19 vaccine rollout

Authors: Li, Chaohua, Douglas, Megan, Zahidi, Rabab, Josiah Willock, Robina, Caplan, Lee, Baltrus, Peter, Gillis, Eric, Mack, Dominic, Gaglioti, Anne

Source: In Preventive Medicine Reports December 2021 24

Effect of Priming With Seasonal Influenza A(H3N2) Virus on the Prevalence of Cross-Reactive Hemagglutination-Inhibition Antibodies to Swine-Origin A(H3N2) Variants

Authors: Liu, Feng, Veguilla, Vic, Gross, F. Liaini, Gillis, Eric, Rowe, Thomas, Xu, Xiyan, Tumpey, Terrence M., Katz, Jacqueline M., Levine, Min Z., Lu, Xiuhua

Source: The Journal of Infectious Diseases, 2017 Sep . 216, S539-S547.

Access URL: https://www.jstor.org/stable/26491578

Cross-Reactive Antibody Responses to Novel H5Nx Influenza Viruses Following Homologous and Heterologous Prime-Boost Vaccination with a Prepandemic Stockpiled A(H5N1) Vaccine in Humans

Authors: Levine, Min Z., Holiday, Crystal, Liu, Feng, Jefferson, Stacie, Gillis, Eric, Bellamy, Abbie R., Tumpey, Terrence, Katz, Jacqueline M.

Source: The Journal of Infectious Diseases, 2017 Sep . 216, S555-S559.

Access URL: https://www.jstor.org/stable/26491580

Scaffold modifications to the 4-(4, 4-dimethylpiperidinyl) 2, 6-dimethylpyridinyl class of HIV-1 allosteric integrase inhibitors

Authors: Parcella, Kyle, Patel, Manoj, Tu, Yong, Eastman, Kyle, Peese, Kevin, Gillis, Eric, Belema, Makonen, Dicker, Ira B., McAuliffe, Brian, Ding, Bo, Falk, Paul, Simmermacher, Jean, Parker, Dawn D., Sivaprakasam, Prasanna, Khan, Javed A., Kish, Kevin, Lewis, Hal, Hanumegowda, Umesh, Jenkins, Susan, Kadow, John F., Krystal, Mark, Meanwell, Nicholas A., Naidu, B. Narasimhulu

Source: Bioorganic & medicinal chemistry. 67

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100164713346.0x000001&indx=1&recIds=ETOCvdc_100164713346.0x000001

The HIV-1 Capsid-Targeted Inhibitor GSK878 Alters Selection of Target Sites for HIV DNA Integration.

Authors: Marquis, Kaitlin A., Everett, John, Cantu, Adrian, McFarland, Alexander, Sherrill-Mix, Scott, Krystal, Mark, Parcella, Kyle, Gillis, Eric, Fridell, Robert A., Bushman, Frederic D.

Source: AIDS Research & Human Retroviruses; Feb2024, Vol. 40 Issue 2, p114-126, 13p

Apparatus and methods for the automated synthesis of small molecules

Synthesis of many different types of organic small molecules using one automated process

Authors: Li, Junqi, Ballmer, Steven G., Gillis, Eric P., Fujii, Seiko, Schmidt, Michael J., Palazzolo, Andrea M. E., Lehmann, Jonathan W., Morehouse, Greg F., Burke, Martin D.

Source: Science, 2015 Mar . 347(6227), 1221-1226.

Access URL: http://www.jstor.org/stable/24746262

Methods for forming protected organoboronic acids

Apparatus and methods for the automated synthesis of small molecules

Automated synthesis of small molecules using chiral, non-racemic boronates

Hepatitis C virus inhibitors

Vinyl MIDA boronate: a readily accessible and highly versatile building block for small molecule synthesis

Authors: Uno, Brice E., Gillis, Eric P., Burke, Martin D.

Source: In Tetrahedron 2009 65(16):3130-3138

Potent Long-Acting Inhibitors Targeting the HIV‑1 Capsid Based on a Versatile Quinazolin-4-one Scaffold.

Authors: Gillis, Eric P., Parcella, Kyle, Bowsher, Michael, Cook, James H., Iwuagwu, Christiana, Naidu, B. Narasimhulu, Patel, Manoj, Peese, Kevin, Huang, Haichang, Valera, Lourdes, Wang, Chunfu, Kieltyka, Kasia, Parker, Dawn D., Simmermacher, Jean, Arnoult, Eric, Nolte, Robert T., Wang, Liping, Bender, John A., Frennesson, David B., Saulnier, Mark

Source: Journal of Medicinal Chemistry; 2/9/2023, Vol. 66 Issue 3, p1941-1954, 14p

Methods for forming protected organoboronic acids

Slow release of organoboronic acids in cross-coupling reactions

System for controlling the reactivity of boronic acids

System for controlling the reactivity of boronic acids

Methods for Forming Protected Organoboronic Acids

Slow Release of Organoboronic Acids in Cross-Coupling Reactions