Multivalent pyrrolidines acting as pharmacological chaperones against Gaucher disease

Authors: Borie-Guichot, Marc, Lan Tran, My, Garcia, Virginie, Oukhrib, Abdelouahd, Rodriguez, Frédéric, Turrin, Cédric-Olivier, Levade, Thierry, Génisson, Yves, Ballereau, Stéphanie, Dehoux, Cécile

Source: In Bioorganic Chemistry May 2024 146

Lipase-catalysed enantioselective kinetic resolution of rac-lipidic alkynylcarbinols and a C5 synthon thereof via a hydrolysis approach

Authors: de Almeida, Diana Kelly Castro, da Silva, Marcos Reinaldo, de Mattos, Marcos Carlos, Nunes, Fátima Miranda, Ballereau, Stéphanie, Génisson, Yves, Maraval, Valérie, Chauvin, Remi, Oliveira, Maria Conceição Ferreira ^*

Source: In Molecular Catalysis June 2020 488

Iminosugar-based ceramide mimicry for the design of new CERT START domain ligands

Authors: Santos, Cécile, Stauffert, Fabien, Ballereau, Stéphanie, Dehoux, Cécile, Rodriguez, Frédéric, Bodlenner, Anne, Compain, Philippe, Génisson, Yves

Source: In Bioorganic & Medicinal Chemistry 15 March 2017 25(6):1984-1989

Ethynylogation approach in pharmacophore design: from alkynyl-to butadiynyl-carbinols vs antitumoral cytotoxicity

Authors: Listunov, Dymytrii, Saffon-Merceron, Nathalie, Joly, Etienne, Fabing, Isabelle, Génisson, Yves, Maraval, Valérie, Chauvin, Remi

Source: In Tetrahedron 20 October 2016 72(42):6697-6704

Extended structural modulation of bio-inspired chiral lipidic alkynylcarbinols as antitumor pharmacophores

Authors: Listunov, Dymytrii, Billot, Chelmia, Joly, Etienne, Fabing, Isabelle, Volovenko, Yulian, Génisson, Yves, Maraval, Valérie, Chauvin, Remi

Source: In Tetrahedron 14 October 2015 71(41):7920-7930

Development of a CERT START Domain–Ceramide HTRF Binding Assay and Application to Pharmacological Studies and Screening

Authors: Fleury, Laurence, Faux, Céline, Santos, Cécile, Ballereau, Stéphanie, Génisson, Yves, Ausseil, Frédéric ^*

Source: In SLAS Discovery July 2015 20(6):779-787

The CERT antagonist HPA-12: First practical synthesis and individual binding evaluation of the four stereoisomers

Authors: Santos, Cécile, Fleury, Laurence, Rodriguez, Frédéric, Markus, Jozef, Berkeš, Dušan, Daïch, Adam, Ausseil, Frédéric, Baudoin-Dehoux, Cécile, Ballereau, Stéphanie, Génisson, Yves

Source: In Bioorganic & Medicinal Chemistry 1 May 2015 23(9):2004-2009

Rapid access to jaspine B and its enantiomer

Authors: Santos, Cécile, Fabing, Isabelle, Saffon, Nathalie, Ballereau, Stéphanie, Génisson, Yves

Source: In Tetrahedron 2 September 2013 69(35):7227-7233

Single- and double-chained truncated jaspine B analogues: asymmetric synthesis, biological evaluation and theoretical study of an unexpected 5-endo-dig process

Authors: Salma, Yahya, Ballereau, Stéphanie, Ladeira, Sonia, Lepetit, Christine, Chauvin, Remi, Andrieu-Abadie, Nathalie, Génisson, Yves

Source: In Tetrahedron 10 June 2011 67(23):4253-4262

Synthesis and biological evaluation of aziridine-containing analogs of phytosphingosine

Authors: Ballereau, Stéphanie, Andrieu-Abadie, Nathalie, Saffon, Nathalie, Génisson, Yves

Source: In Tetrahedron 2011 67(14):2570-2578

Ionic Liquids and the Heck Coupling Reaction: An Update

Authors: Prediger, Patricia, Genisson, Yves, Roque Duarte Correia, Carlos

Source: Current organic chemistry. 17(3):238-256

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100083471500.0x000001&indx=1&recIds=ETOCvdc_100083471500.0x000001

Alteration of Ceramide 1-O-Functionalization as a Promising Approach for Cancer Therapy

Authors: Ballereau, Stephanie, Levade, Thierry, Genisson, Yves, Andrieu-Abadie, Nathalie

Source: Anti-cancer agents in medicinal chemistry. 12(4):316-328

Availability: http://explore.bl.uk/primo_library/libweb/action/display.do?tabs=detailsTab&gathStatTab=true&ct=display&fn=search&doc=ETOCvdc_100083462100.0x000001&indx=1&recIds=ETOCvdc_100083462100.0x000001

The natural marine anhydrophytosphingosine, Jaspine B, induces apoptosis in melanoma cells by interfering with ceramide metabolism

Authors: Salma, Yahya, Lafont, Elodie, Therville, Nicole, Carpentier, Stéphane, Bonnafé, Marie-José, Levade, Thierry, Génisson, Yves, Andrieu-Abadie, Nathalie

Source: In Biochemical Pharmacology 1 September 2009 78(5):477-485

Synthesis and biological evaluation of conformationally constrained analogues of the antitubercular agent ethambutol

Authors: Faugeroux, Vanessa, Génisson, Yves, Salma, Yahya, Constant, Patricia, Baltas, Michel

Source: In Bioorganic & Medicinal Chemistry 2007 15(17):5866-5876

New approach to carbamoyl-polyoxamic acid derivatives through an oxazolidinone synthon

Authors: Collet, Magalie, Génisson, Yves, Baltas, Michel

Source: In Tetrahedron: Asymmetry 2007 18(11):1320-1329

Enantioselective access to a versatile 4-oxazolidinonecarbaldehyde and application to the synthesis of a cytotoxic jaspine B truncated analogue

Authors: Génisson, Yves, Lamandé, Lydia, Salma, Yahya, Andrieu-Abadie, Nathalie, André, Chantal, Baltas, Michel

Source: In Tetrahedron: Asymmetry 2007 18(7):857-864

N,O-Dialkyl deoxynojirimycin derivatives as CERT START domain ligands

Authors: Castellan, Tessa, Santos, Cécile, Rodriguez, Frédéric, Lepage, Mathieu L., Liang, Yan, Bodlenner, Anne, Compain, Philippe, Génisson, Yves, Dehoux, Cécile, Ballereau, Stéphanie

Source: In Bioorganic & Medicinal Chemistry Letters 15 January 2020 30(2)

New chiral imidazolinic derivatives

Authors: Génisson, Yves, Viguerie, Nancy Lauth-de, André, Chantal, Baltas, Michel, Gorrichon, Liliane

Source: In Tetrahedron: Asymmetry 7 March 2005 16(5):1017-1023

This result is not displayed to guests.
Login for full access.

This result is not displayed to guests.
Login for full access.